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6-{3-oxo-3-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
6-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyrazine-2-carboxamide
1-[(4-chlorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylbenzamide
4-{3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
8-(3,5-dimethyl-1H-pyrazol-4-yl)quinoline
1-methyl-3-propyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-[2-(pyrrolidin-1-yl)ethyl]piperazine
[5-(1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
2-amino-4-(3-ethenylphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-[3-methyl-4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H-pyrazolo[3,4-d]imidazol-5-yl)-1H-pyrazol-1-yl]ethan-1-ol
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-N-ethylpyrimidin-2-amine
4-(2-methylpyridine-3-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-4-amino-N,N-diethyl-1-(4-fluoro-2-methylbenzenesulfonyl)pyrrolidine-2-carboxamide
N-cyclopropyl-4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazine-2-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,2-dimethylpropanamide
3-methyl-4-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)amino]-N-propylbenzamide
3-phenyl-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-ol
3-(3-chlorophenyl)-N-cyclopropyl-3-(3-hydroxyphenyl)propanamide
2-methoxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(furan-3-ylmethyl)-4-(pyridin-2-ylmethyl)piperazine
2-[2-(furan-3-yl)-4-methylphenoxy]acetamide
1-[5-({[(2-chlorophenyl)methyl]sulfanyl}methyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]butan-2-ol
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
3-benzyl-5-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1H-1,2,4-triazole
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(1-cyclobutanecarbonylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-N'-methyl-N'-phenylethanediamide
1-benzyl-6-(pyridin-3-ylmethoxy)-4-(quinolin-5-ylmethyl)-1,4-diazepan-2-one
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
6-[3-(pyridin-3-yl)azetidin-1-yl]pyridine-3-carbonitrile
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-[2-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
5-(2-{4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
N1-(3-methylpyridin-4-yl)-N2-[4-(pyridin-2-yl)pyrimidin-2-yl]ethane-1,2-diamine
5-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}quinoxaline
(1R,5S,6S)-6-{[4-(3,4-dichlorophenyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-[(4aR,7aS)-6,6-dioxo-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
5-acetamido-2-ethyl-N-[(4-fluorophenyl)methyl]-N-methyl-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
2-{5-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
8-(3-methylpyrazin-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-methyl-3-{7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)methanesulfonamide
7-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(5-chloro-2-methylphenyl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
2-(2H-1,2,3-benzotriazol-2-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
2-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]-4,6-bis(propan-2-yl)phenol
N-[3-({[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide