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2,3-dimethyl-6-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(3-methoxyphenoxy)propan-1-one
(4aR,7aS)-1-(2-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]pyridine-4-carboxamide
7-(2-methoxyethyl)-2-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
N-benzyl-N-methyl-3-(morpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[(1S,3S,3aR,6aS)-5-ethyl-3-(hydroxymethyl)-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-4-fluorophenol
1-(difluoromethyl)-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
2,4-dimethyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
7-(3,6-dimethylpyrazin-2-yl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,7aR)-1-(2-methoxy-3-methylbenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1,3-thiazole-4-carboxamide
1-({5-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,4-difluoropiperidine
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-(3-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)acetamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(pyrrolidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-5-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}phenol
{[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}(thiophen-3-ylmethyl)amine
3-(2,3-dimethylphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
(4S)-3-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
(4aS,8aR)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(benzenesulfonyl)piperazin-1-yl]propan-1-one
N-tert-butyl-3-[2-(5-acetamido-1H-1,2,4-triazol-3-yl)acetamido]-2-methylbenzamide
8-fluoro-3-{4-[2-(2-hydroxyethoxy)ethyl]piperazine-1-carbonyl}-1,4-dihydroquinolin-4-one
N-[(3R,4R)-3-hydroxy-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl]pyridine-4-carboxamide
N,N-dimethyl-2-{[3-(pyridin-2-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-cycloheptyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
2-hydroxy-1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(methylsulfanyl)butan-1-one
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(quinolin-8-ylmethyl)amine
2-(2-chlorophenyl)-N-(cyclopropylmethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(3-methylpyridine-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidine-3-carbonyl]-4-(pyridin-2-yl)piperidin-4-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(1,3-dihydroxypropan-2-yl)acetamide
3-{2-[4-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
6-methoxy-N,3-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1-benzofuran-2-carboxamide
3-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
N-{1-oxaspiro[4.4]nonan-3-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(adamantan-1-ylmethyl)-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}pyrrolidine-1-carboxamide
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]butane-1,2-dione
3-[(2-fluorophenyl)formamido]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
5-{4-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
N-{1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]piperidin-4-yl}methanesulfonamide