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4-(2-{2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)morpholine
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-ol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(dimethylamino)-2,2-dimethylpropyl]acetamide
5-methanesulfonyl-1'-(oxolan-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclohexyl-2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
2-(2-chloro-4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)propanoic acid
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(3R,4S)-1-[(3-ethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-acetyl-N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
4-(3,4-dimethylbenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(4-chloro-2,5-dimethylbenzenesulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(naphthalen-1-ylmethyl)-1,2-oxazole-3-carboxamide
7-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
3,4-dichloro-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
methyl[(5-methyl-1H-indol-3-yl)methyl](oxan-2-ylmethyl)amine
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-4-methylpyrimidin-2-amine
3-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
(3S,4R)-4-(2-methylphenyl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
2-({[(furan-2-ylmethyl)carbamoyl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-[2-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-2-yl)ethyl]phenol
methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-(cyclopropylmethyl)-N-(2-methoxyethyl)-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[(2S)-1-methylpyrrolidine-2-carbonyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-3-methanesulfonyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-{2-[(pyridin-3-yl)amino]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-6-(propan-2-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-4-amine
8-(1H-indol-3-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}ethyl)-4-methylpiperazine
7-methoxy-N,N-dimethyl-2-[2-(morpholin-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(4H-1,2,4-triazol-4-yl)benzamide
4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-(1-methyl-1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-({1-azabicyclo[2.2.2]octan-3-yl}amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-[1-(2,6-dimethylquinolin-4-yl)-N-methylformamido]-2-(pyridin-3-yl)acetic acid
1'-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-5-methoxy-1,4-dihydropyridin-4-one
2-(2,5-dimethoxyphenyl)-N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2,5,7-trimethyl-4-[3-(morpholin-4-yl)piperidine-1-carbonyl]quinoline
2-(butane-1-sulfonamidomethyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid