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3-methyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
5-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-{1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperidin-4-yl}-1,3-benzoxazole
N-[2-(pyrrolidin-1-yl)ethyl]quinoxaline-5-carboxamide
2-ethyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
1-ethyl-4,6-dimethyl-2-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2-dihydropyridine-3-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{5-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]-2-methylphenyl}imidazolidin-2-one
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N,N-dimethylpyridin-2-amine
N4-({2-[(dimethylamino)methyl]phenyl}methyl)-N4,6-dimethylpyrimidine-2,4-diamine
2-[4-(aminomethyl)piperidine-1-carbonyl]-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
4-methoxy-N-({1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
3-(hydroxymethyl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-ol
2-[4-(5-aminopyrazin-2-yl)-1H-pyrazol-1-yl]-N-(1-benzyl-1H-pyrazol-3-yl)acetamide
2-methyl-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
N-cyclohexyl-N-methyl-3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyridin-2-amine
(3R,4S)-4-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-oxo-4-phenylbutanamide
N-[(5-ethylpyridin-2-yl)methyl]-3-[(2-fluorophenyl)formamido]-N-methylpropanamide
6-methyl-2-{1-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
N-[(1-ethylpyrrolidin-3-yl)methyl]-4-methoxy-2,3,6-trimethylbenzene-1-sulfonamide
N-(3-ethylphenyl)-1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
6-{[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}naphthalen-2-ol
2-ethyl-6-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-[(diethylamino)methyl]-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(benzyloxy)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]butanamide
1-[1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrrolidin-2-one
2-ethoxy-5-{2-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
1-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-3-phenylpyrrolidin-3-ol
5-(furan-3-yl)-1-(3-methylbutan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methylpiperidin-4-amine
2-(2-methylpropyl)-4-[6-(propan-2-yl)pyrimidin-4-yl]morpholine
2-methyl-4-(5-{[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
7-(propan-2-yl)-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(2,4-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,2R,6S,7S)-4-(3-chlorothiophene-2-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyridin-3-ol
N-(1,2,3-thiadiazol-5-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
3-(2-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
1-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
N-benzyl-4-(4-{[(3R)-3-hydroxypiperidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide