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3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
4-(2-methoxy-5-methylphenyl)-3-(oxan-4-yl)-4H-1,2,4-triazole
1-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)imidazolidine-2,4-dione
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
2-(2-{[4-(propan-2-yl)piperidin-1-yl]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
2-fluoro-N-({3-methyl-7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(3-methoxyphenyl)urea
(1S,5R)-6-(2-methoxyethyl)-3-(4-methylpyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-cyclobutyl-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3,4-oxadiazol-2-amine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]methyl}pyridine
3-(3-methoxyphenoxy)-1-{[3-(methylsulfanyl)phenyl]methyl}azetidine
7-chloro-4-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}quinolin-2-amine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(quinazolin-4-yl)piperazin-1-yl]acetamide
(2S,4S,5R)-2-ethyl-4-[(2-hydroxyethyl)(methyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-(3-chlorophenyl)-4-[4-(1H-imidazol-1-yl)benzoyl]piperazin-2-one
2-{[(1-methyl-1H-imidazol-2-yl)methyl](propyl)amino}-N-(1,3-thiazol-2-yl)propanamide
2-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]morpholin-3-yl}-1-(thiomorpholin-4-yl)ethan-1-one
2-(furan-2-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
(2E)-N-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-3-phenylprop-2-enamide
2-{[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
3-({[1-(4,7-dimethylquinazolin-2-yl)azepan-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
(2R,3R)-3-{[2-(1H-indol-1-yl)ethyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-cyclopropyl-8-[2-(pyrrolidin-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}(pyridin-2-ylmethyl)amino)butan-1-ol
N-[2-(dimethylamino)ethyl]-1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(2-methoxyphenoxy)ethan-1-one
ethyl 1-[(3-{[1-(thiophene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
4-(6-chloro-2H-chromen-3-yl)-7-hydroxy-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(2-chlorophenyl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-(5-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-(1-benzothiophen-2-ylmethyl)-1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
N-(2,3-dihydroxypropyl)-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
3-{2-oxo-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
4-{[4-(ethanesulfonyl)piperazin-1-yl]methyl}-6-ethyl-2H-chromen-2-one
(3S,4R)-1-(7-chloro-1-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
3-{2-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-(2H-1,3-benzodioxol-5-yl)-1-(1-methylpiperidin-4-yl)-1-(pyridin-4-ylmethyl)urea
3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
4-(2-benzyl-3-oxopiperazine-1-carbonyl)-1-methyl-1,2-dihydroquinolin-2-one
4-{[2-hydroxy-5-(6-methoxypyridin-2-yl)phenyl]methyl}piperazine-1-carbaldehyde
4-[(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)methyl]benzamide
4-methoxy-6-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-benzyl-N-methyl-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide