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1-[4-(pyrrolidine-1-carbonyl)benzenesulfonyl]-1,4-diazepan-5-one
1-{[5-(1-ethylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
ethyl 2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-1,3-oxazole-4-carboxylate
3-[2-({[1-(4-fluorophenyl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-N-cyclopropylpiperazine-2-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-3-azaspiro[5.5]undecan-9-amine
3-{1-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-(2-{furo[3,2-c]pyridin-4-yl}-5-methoxyphenyl)-1H-pyrazole
4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}thiomorpholine
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
8-[(2-chloro-6-fluorophenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-tert-butylphenoxymethyl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
ethyl 4-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
2-acetyl-8-[(4-hydroxy-3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-phenyl-1,2,4-oxadiazole
ethyl (4aS,8aR)-6-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylate
4-[3-(hydroxymethyl)-4-propoxyphenyl]-N,N-dimethylbenzamide
1-[2-(dimethylamino)ethyl]-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
8-[(4-acetylphenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(4-phenyl-1H-1,2,3-triazol-1-yl)-1-(1-propylpiperidin-4-yl)piperidine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-6-(2-hydroxypyridine-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
methyl 2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidine-1-carboxylate
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{[2-(methoxymethyl)piperidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
2-{1-cyclohexyl-5-[(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
3-({[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
methyl 3-{[(3-chlorophenyl)formamido]methyl}-5-(furan-2-amido)benzoate
2-(5-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
1-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
5-methyl-4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
3-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
{[5-(furan-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
2-[(4aR,7aS)-4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-(2-ethoxyethyl)-N-methyl-N-(oxan-4-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(cyclohex-3-en-1-ylmethyl)methylamine
1-methyl-1-[(2-methylpyridin-4-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
4-[2-(4-fluorophenyl)morpholine-4-carbonyl]pyridin-3-ol
4-methyl-2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-methyl-6-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}pyrimidin-4-amine
4-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-2-(propan-2-yl)-1,3-oxazole
5-(2-chlorophenyl)-4-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-3-yl]pyrimidine
8-fluoro-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}quinoline-2-carboxamide
N-cyclopropyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
6-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide