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3-(5-methylthiophen-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-methylbut-2-en-1-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-3-carboxamide
3-{[(5-fluoro-2-hydroxyphenyl)methyl](propan-2-yl)amino}propanamide
5-{[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,3-oxazolidin-2-one
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-5-oxo-5-phenylpentanamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
4-{[(2-amino-5-ethylpyrimidin-4-yl)amino]methyl}-N,N-dimethylbenzamide
7-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
3-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[4-(difluoromethoxy)-2-methylphenyl]urea
N-({1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
2-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2,3,4-tetrahydroquinoline-6-sulfonamide
N-methyl-4-(morpholin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide
3-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(thiophene-2-carbonyl)piperidine
2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
8-[(4-chloro-3-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropanecarbonyl-1'-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-fluorophenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}methanesulfonamide
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(2,3-dihydro-1H-inden-4-yl)urea
methyl (2S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-acetamidopyrrolidine-2-carboxylate
2-(1-benzyl-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-{5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2-methylphenyl}oxolane-2-carboxamide
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
N-[3-oxo-3-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propyl]acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-(2-oxopyrrolidin-1-yl)benzamide
(2S)-3-(4-hydroxyphenyl)-2-{imidazo[1,2-a]pyridin-6-ylformamido}propanamide
N3-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[2-(3-chlorophenoxy)propanoyl]-1-ethyl-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl (2S)-2-{[1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
1-{3-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-(3-aminopropyl)-3-(2-chlorophenyl)-3-phenylpropanamide
(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-(hydroxymethyl)piperidine-1-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
3,3-dimethyl-1-({5-[(2-propoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
3-(3-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
3-(azepane-1-carbonyl)-5-[4-(2-methoxyethyl)piperazin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole
{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}methanamine
4-[(1S,2R)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-hydroxypropyl]phenol
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]propanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrazine-2-carboxamide
4-(3-chlorophenoxy)-1-[2-(3-methyl-1,2-oxazol-5-yl)ethyl]piperidine
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-[(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl)methyl]-1H-indole-2-carboxamide