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N-cyclohexyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-3-(pyridin-4-yl)propanamide
[(3R,4R)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(1R,5S)-3-benzyl-6-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1-benzothiophene-5-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanamide
(2S,4S)-4-amino-N-ethyl-1-(1H-indol-4-ylmethyl)pyrrolidine-2-carboxamide
[(2R)-1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
N-ethyl-3-(3-hydroxyquinoxalin-2-yl)-N-(oxan-4-ylmethyl)propanamide
8-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-(cyclohex-3-ene-1-carbonyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-2-{3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}azepane
3-[(2-chloro-5-acetamidophenyl)formamido]-N-(2-ethylphenyl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-[(3-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-3-ethoxypropanamide
4-[5-(5-fluoro-3-methyl-1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]butan-2-ol
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-[(2,3-difluorophenyl)methyl]piperazin-2-one
1-[4-(aminomethyl)piperidin-1-yl]-3-(azocan-1-yl)propan-1-one
4-(2-butyl-1H-imidazol-4-yl)-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
2-cyclopropyl-N-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-2-ylmethyl)piperidin-2-one
methyl 6-(3-{2-[(5-chloro-2-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)pyridine-3-carboxylate
2-(8-methoxy-2-methylquinolin-5-yl)benzamide
8-(2-ethoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(8-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]benzamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-methyl-1H-indazole-3-carboxamide
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(2-phenoxyethyl)piperazine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4-trimethoxybenzamide
4-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
1-{2-[(3,4-dimethoxyphenyl)formamido]ethyl}-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}pyridin-3-ol
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[(3S)-2-oxoazepan-3-yl]piperidine-4-carboxamide
3-{5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
4-ethyl-6-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrimidine
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
1-[(4-fluorophenyl)methyl]-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-(morpholin-3-yl)acetamide
2-(2-chlorophenyl)-N-[3-(dimethylamino)propyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-(4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
3-[2-(diethylamino)-2-(furan-2-yl)ethyl]-1-(4-oxo-4H-chromen-6-yl)urea
N-(1-phenylethyl)-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
1-(4-methoxy-3-methylphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(1R,2S,9R)-11-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-propyl-1,3-thiazole-4-carboxamide