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3-(azepane-1-carbonyl)-N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,5R)-N-(6-methylpyridin-3-yl)-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
methyl 4-[(3-{2-[(2-fluorophenyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
3-[3-(4-hydroxyphenyl)propanoyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
2-ethyl-9-(2-methoxyacetyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
8-(1,3-benzothiazol-2-ylmethyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl({[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl})[1-(pyridin-2-yl)propan-2-yl]amine
4-{4-[(5-chlorothiophen-2-yl)methyl]piperazin-1-yl}-2-methyl-6-(propan-2-yl)pyrimidine
N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[1-(thiophen-2-yl)ethyl]acetamide
1-(2-methoxyethyl)-4-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]pyrrolidin-2-one
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-phenylpiperazin-2-one
2-(2-chlorophenyl)-N-ethyl-N-(2-methoxyethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(carbamoylmethyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)piperidine-3-carboxamide
N-[4-(butan-2-yl)phenyl]-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetamide
[(3R,4R)-1-cyclobutanecarbonyl-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-[(3-methoxyphenyl)methyl]-4-(3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazin-2-one
(1R,5R)-3-cyclobutanecarbonyl-6-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-aminopyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
4-{3-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}morpholine
N-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-ylmethyl)piperidin-3-amine
2-(4-tert-butylphenyl)-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}acetic acid
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
2-methoxy-5-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazin-1-yl]methyl}pyrimidine
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(4aR,7aS)-1-ethyl-4-[2-(morpholin-4-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-({1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropyl}methyl)-1H-pyrazole
4-[2-(cyclopentyloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
9-(2,3-difluoro-4-methoxybenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-4-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}butanamide
2-(3-methylphenyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(2-hydroxyethyl)-3-[5-(1H-indol-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
2-methyl-8-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
(3S,4S)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
5-(piperidin-1-yl)-2-[(2,4,5-trifluorophenyl)methyl]-2,3-dihydropyridazin-3-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
3-(1H-1,3-benzodiazol-2-ylmethyl)-N-benzylpiperidine-1-sulfonamide
4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
2-[(2-ethylpiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
(1R,3S)-3-methoxy-7-[2-(morpholin-4-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
2,6-dimethoxy-3-(3-methoxypiperidine-1-carbonyl)pyridine
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-5-methylthiophene-2-carboxamide
N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(pyrimidin-4-ylmethyl)acetamide