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1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
5-methoxy-2-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-[(3R,4S)-4-(3-methoxyphenyl)-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidin-3-yl]acetamide
N-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
8-(3-fluoro-4-methylbenzenesulfonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)thiophene-2-carboxamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
N-[2-(4-hydroxyphenyl)ethyl]-2-[4-(1-methyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]acetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-(4-ethoxy-3-methylphenyl)-4-oxo-N-[3-(pyrrolidin-1-yl)propyl]butanamide
2-amino-6-cyclopentyl-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-ethyl-N-(2-hydroxyethyl)acetamide
1-(4-methyl-2-{[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amino}pyrimidin-5-yl)ethan-1-one
2-amino-4-[5-(oxolan-2-yl)thiophen-2-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2-[(2-{ethyl[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
ethyl 1-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}piperidine-2-carboxylate
3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}pyridine
(2R,6R)-4-[5-(methoxymethyl)thiophene-2-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3R,4S)-4-[({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(ethyl)amino]oxolan-3-ol
4-[(2-methoxypyrimidin-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-[(2-methylphenyl)methyl]piperidin-3-yl)methanol
dimethyl[(4-methyl-5-{1-[1-(4-methylphenyl)piperidin-4-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-4-(piperidin-1-yl)butanamide
2-(2-{[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-[(4-chlorophenyl)methyl]-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(1H-indol-5-ylmethyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-phenoxypiperidine-4-carboxylic acid
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-6-oxo-1,6-dihydropyridine-2-carboxamide
2-[1-(ethylcarbamoyl)pyrrolidin-3-yl]benzoic acid
6-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyrazine-2-carboxamide
4-benzyl-3-[1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-N,N-diethyl-1-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
7-(1-benzothiophen-3-yl)-4-(1H-imidazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{3-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}propanamide
3-{5-[2-(1H-1,3-benzodiazol-2-ylmethoxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(3R,4S)-1-[2-chloro-5-(piperidin-1-yl)benzoyl]-4-cyclopropylpyrrolidin-3-amine
2-(ethanesulfonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-ethyl-5-[3-(1H-imidazol-1-yl)propyl]-1,3-benzoxazole
4-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
4-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]azetidin-3-yl}morpholine
2-{2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]ethyl}-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
(2R)-2-[5-(3-chloro-4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
1-[5-(quinolin-8-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
3-[5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
11-{[(2,4-difluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(2-methylquinolin-8-yl)-3-[2-(propane-2-sulfonyl)ethyl]urea
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one