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3-{[(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
3,5-dimethoxy-2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)benzoic acid
N-[(3-ethoxy-4-methoxyphenyl)methyl]-2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}methyl)-6,8-dimethylquinolin-4-ol
3-[(3R,4S)-4-(morpholin-4-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]propan-1-ol
N-butyl-2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(3-methoxyphenyl)methyl]acetamide
4,6-dimethyl-1-{3-[2-(2-methylphenyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2-dihydropyrimidin-2-one
N-(cyclohex-1-en-1-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
2-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
3-[(4aR,7aS)-4-{2-[(dimethylcarbamoyl)amino]acetyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-(propan-2-yl)-1-(2-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(3-methoxypropanoyl)piperidine-3-carboxamide
2-(3-chlorophenoxymethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
2-(2,5-dioxoimidazolidin-4-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-fluorobenzamide
9-methoxy-7-(3-methoxyphenyl)-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(oxan-2-ylmethyl)amino]pyridine-3-carboxamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
5-[1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-2-one
3-(2-ethoxypyridin-3-yl)-5,6-dimethyl-1,2-dihydropyridin-2-one
3-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)benzonitrile
(3S,5R)-5-(cyclopropylcarbamoyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-3-carboxylic acid
N-butyl-6-oxo-N-(thiophen-3-ylmethyl)-1,6-dihydropyridine-2-carboxamide
3-(3-chlorophenyl)-3-phenyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]propanamide
(1S,5R)-6-benzyl-3-(thiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-5-propylpyrimidine
4-{[2-(1H-pyrrol-1-yl)ethyl]sulfamoyl}-N-[(3R)-pyrrolidin-3-yl]benzamide
8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-fluoro-2-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)quinolin-4-ol
4-ethyl-1-methyl-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(6-methylpyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{2-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}pyrrolidine
5-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
ethyl (4aS,8aR)-6-(2-amino-9H-purin-6-yl)-decahydro-1,6-naphthyridine-4a-carboxylate
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[({3-[(furan-2-ylmethyl)sulfanyl]propyl}amino)methyl]piperidin-3-ol
3-benzyl-1-methyl-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4,6-dimethoxy-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[5-(2-ethylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-1-[3-(pyridin-2-yl)propyl]urea
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-phenyl-1,4-diazepane
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one