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6-oxo-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}piperazine-2-carboxamide
2-methoxy-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
3-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1,2-dihydrophthalazin-1-one
2-(3-phenylpropyl)-N-[2-(pyrazin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
(4aS,8aR)-6-(cyclopent-3-en-1-yl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-2-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)acetamide
1-methyl-4-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
N-(butan-2-yl)-3-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-4-phenylpyrimidin-2-amine
1-(furan-2-ylmethyl)-4-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]piperidine
4-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
4,6-dimethyl-3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
3-(4-hydroxyphenyl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(3aS,6aS)-5-{[4-(difluoromethoxy)phenyl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-(benzyloxy)butan-1-one
N-(2-hydroxyethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
2-methyl-5-({4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}methyl)pyrazine
1-{2-[1-(2,3-dihydro-1H-inden-4-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
methyl({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-({1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopropanecarboxamide
2-methoxy-N-[(3R,4S)-4-(3-methoxyphenyl)-1-(oxan-4-yl)pyrrolidin-3-yl]acetamide
1-cyclopentanecarbonyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
N-(2-methyl-1-benzofuran-5-yl)-4-(thian-4-yl)piperazine-1-carboxamide
4-(4-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
3-{4-[2-(azepan-1-yl)acetyl]piperazin-1-yl}pyrazine-2-carbonitrile
(2S,4S)-4-amino-N,N-diethyl-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)pyrrolidine-2-carboxamide
3-cyclopropyl-N-(5-methyl-1,2-oxazol-3-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazole-5-carboxamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-[2-(pyrrolidin-1-yl)ethyl]pyridin-2-amine
1-methyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
2,2-dimethylpropyl 3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
5-methoxy-2-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-4H-pyran-4-one
N-cyclobutyl-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-(1,2-oxazinane-2-carbonyl)-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
1-[1-(3-chloro-5-fluorobenzoyl)piperidin-4-yl]-3-methylbutan-1-ol
1-[(2-fluorophenyl)methyl]-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
2-(3-ethoxyphenyl)-5-(pyrrolidine-1-carbonyl)pyridine
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
ethyl 4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(methylsulfanyl)pyrimidine-5-carboxylate
[(4aS,8aR)-6-{7-amino-2-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
5-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-2-(naphthalen-2-yl)pyrimidine
(3S,4S)-4-methyl-1-[5-(morpholin-4-ylmethyl)pyridin-2-yl]piperidine-3,4-diol
(1S,5R)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
2-[4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
7-fluoro-2-methyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}quinoline-4-carboxamide
N-methyl-4-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine