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(2S,4R)-4-{4-[2-(2-cyclopentylacetamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
1-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1H-1,2,4-triazole
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(2-phenoxyethyl)piperazine
7-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({4-hydroxy-1-[(6-methoxy-2H-chromen-3-yl)methyl]azepan-4-yl}methyl)acetamide
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
2-amino-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
N-(6-methyl-2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-cyclopropyl-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[2-(trifluoromethyl)phenyl]urea
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(pyridin-2-yl)pyrimidine
1-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzenesulfonyl}piperazine
3-(5-ethyl-4H-1,2,4-triazol-3-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]aniline
3,5-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
[1-(5-amino-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
1-(4-fluorophenyl)-N,2,2-trimethyl-N-[(3-methyl-1H-indol-2-yl)methyl]cyclopropane-1-carboxamide
3-hydroxy-3-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)-1-(2-methoxyethyl)piperidin-2-one
N-{3-[6-(piperidine-1-carbonyl)pyrazin-2-yl]phenyl}acetamide
4-(piperidine-1-carbonyl)-2-(pyridin-4-yl)pyridine
N-[1-(4-methanesulfonylphenyl)propyl]-5-(methoxymethyl)furan-2-carboxamide
(1S,4R)-4,7,7-trimethyl-3-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-2-oxabicyclo[2.2.1]heptane-1-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
2-methyl-1-{[3-(2-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole
9-[2-(1H-imidazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[1-(piperidin-1-yl)cyclopentyl]methyl}pyrrolidin-2-one
7-[(2-fluorophenyl)methyl]-2-(5-methyl-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-tert-butyl-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
7-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1'-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-(oxan-4-yl)-3,4-dihydropyrimidin-4-one
2-fluoro-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-sulfamoylbenzamide
5-(1-{[3-(pyrimidin-2-yloxy)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-[(1-benzyl-3-methyl-1H-1,2,4-triazol-5-yl)(pyridin-3-yl)methyl]morpholine
4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(1,3-thiazole-5-carbonyl)piperidine
1-[(3-fluorophenyl)methyl]-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
7-[2-(2-chlorophenoxy)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-(2-fluoroethyl)-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(1-{[4-(difluoromethoxy)phenyl]methyl}-4-(2-phenylethyl)piperidin-4-yl)methanol
1-(oxan-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine-3-carboxamide
2-methyl-4-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine
1-(2-{[(3-chloro-4-propoxyphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
(1S,5R)-3-benzyl-6-(pyridazine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-ethyl-4-[3-(propoxymethyl)pyrrolidin-1-yl]pyrimidin-2-amine
5-({2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1-methylpyrrolidin-2-one
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)acetamide
3-methyl-8-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})(pyrazin-2-ylmethyl)amine