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N-ethyl-5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyrimidin-2-amine
N-benzyl-3-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
2-[2-(dimethylamino)ethyl]-8-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(2S)-3-(1H-imidazol-4-yl)-1-oxo-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-2-yl]acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propan-1-one
1-(cyclobutylmethyl)-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
2-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2-chloro-6-methoxyphenoxy)acetamide
1-(1H-pyrazole-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-(4H-1,2,4-triazol-4-yl)naphthalene-1-carbonitrile
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol
1-{4-[5-(azepane-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
N-[2-cyclobutyl-1-methyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]oxolane-2-carboxamide
[(1-{1-[(6-fluoro-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
3-cyclopropyl-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
(1S,2S)-2-{[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]amino}cyclohexan-1-ol
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[(prop-2-en-1-yl)amino]benzamide
diethyl[(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]amine
2-{4-chloro-2-[1-(oxan-2-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2,3-dihydro-1H-inden-2-yl)-N-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-amine
2-{9-[(4-acetamidophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carbonitrile
2-methyl-3-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoxaline
2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N,N-dimethylacetamide
2-(1H-indol-1-yl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(4aS,7aR)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
dimethyl(2-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)amine
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
2-[(furan-3-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-2-methylphenyl]-2-methylpropanamide
(3S,4S)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
7-methoxy-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1-benzofuran-2-carboxylic acid
ethyl 4-{[4-({1-[3-(trifluoromethyl)benzenesulfonyl]piperidin-3-yl}methoxy)phenyl]methyl}piperazine-1-carboxylate
6-methyl-3-{[4-(pyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-5,6-dihydro-1,4-dioxine-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(2-methylphenyl)-1,3-thiazole
N-(4-{1-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1H-imidazol-2-yl}phenyl)acetamide
3-methyl-2-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-indole
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(2S,4S)-4-amino-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(4-methoxybenzoyl)piperazine
(3aS,6aS)-1-oxo-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
3-(2-{[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(1H-imidazol-1-yl)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide