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N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
6-[(diethylamino)methyl]-N-(pyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1,2-oxazol-3-ylmethyl)-5-[1-(1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-(2-hydroxy-4-methylbenzoyl)piperidin-4-yl]pyridine-3-carboxamide
ethyl 4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazine-1-carboxylate
2-({3-[(2,2-difluoroacetamido)methyl]pyrrolidin-1-yl}methyl)benzoic acid
(1S,2R)-N1-[3-(2-oxopyrrolidin-1-yl)propyl]-N2-propylcyclohexane-1,2-dicarboxamide
N-[3-(furan-2-amido)-4-methoxyphenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
3-(naphthalen-1-yl)-5-(thian-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-propyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
(1S,2S)-2-{[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}cyclohexan-1-ol
(2S)-2-(2,3-difluorophenyl)-2-[2-(1-ethylpiperidin-4-yl)acetamido]acetic acid
3-[(4-{[(5-amino-1H-1,2,4-triazol-3-yl)methyl]amino}-6-methylpyrimidin-2-yl)amino]phenol
methyl 2-({3-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-5-(phenylsulfamoyl)phenyl}formamido)acetate
N,3,5-trimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]furan-2-carboxamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-[4-(morpholine-4-carbonyl)phenyl]thiolan-3-amine
(3S,9aR)-3-benzyl-8-[(2,5-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(4-{4-[(oxolan-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)methyl]-1H-pyrazole-3-carboxylic acid
5-[4-(2-aminopyrimidin-4-yl)piperidine-1-carbonyl]-4-methylpyrimidin-2-amine
3-(2-oxo-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)benzonitrile
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}pyrrolidin-2-one
[1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanol
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[(4-sulfamoylphenyl)methyl]urea
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
8-(1H-1,3-benzodiazole-5-carbonyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(5-methylpyrazine-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-oxo-1,2-dihydroquinoline-3-carboxamide
9-(5-chloropyrimidin-2-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-(3-chlorobenzenesulfonyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
2-(2,5-dioxoimidazolidin-4-yl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}acetamide
5-cyclopropyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
5-ethyl-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
11-{[(2,5-difluorophenyl)methyl]amino}-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-(azepane-1-sulfonyl)-5-[2-(propan-2-yl)-1H-imidazol-1-yl]benzoic acid
N-[(3S,4R)-1-(4-fluoro-2-methylbenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[3-(1H-pyrazol-1-yl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(5-chloro-2-propoxyphenyl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,5S)-N-{2-[4-(dimethylamino)phenyl]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-[(2S)-2-aminobutanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-(azepane-1-carbonyl)-N-(1-benzylpiperidin-4-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine