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1-(2-methoxyphenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazole-4-carboxamide
6-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
2-(1H-1,3-benzodiazol-2-yl)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
1-[cyclopropyl(pyridin-2-yl)methyl]-1-methyl-3-(2-methyl-1-benzofuran-7-yl)urea
6-(2-methoxyethyl)-2-[4-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-benzyl-3-ethyl-1-(2-hydroxypyridine-3-carbonyl)-1,4-diazepan-5-one
1-(2-chlorophenyl)-3-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
4-{2-[2-(2,5-dimethylphenyl)-1H-imidazol-1-yl]-1-(pyridin-4-yl)ethyl}morpholine
2-({4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazol-1-yl}methyl)-1H-indole
4-(4-ethoxy-3-methylphenyl)-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)butanamide
1-[4-(furan-2-yl)phenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
methyl 4-(methylsulfanyl)-2-({[2-(pyridin-3-ylmethoxy)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}amino)butanoate
7-fluoro-2-methyl-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]quinoline-4-carboxamide
3-[5-(4-hydroxy-3,5-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
3-(1H-pyrazol-4-yl)-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
5-(3-oxo-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propyl)imidazolidine-2,4-dione
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-{[3-(3-methoxyphenoxymethyl)piperidin-1-yl]methyl}pyridine
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-hydroxy-3-[2-methoxy-4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-{4-[4-(4-methoxyphenyl)butanoyl]-2-oxopiperazin-1-yl}benzonitrile
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-methyl-3-(2-methylpropyl)-N-(1,2-oxazol-5-ylmethyl)-1,2-oxazole-5-carboxamide
4-(5-fluoro-3-methyl-1H-indol-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]-1-(4-methoxyphenyl)-1H-imidazole
2-(4-fluorophenyl)-1-[(3,4,5-trimethoxyphenyl)methyl]azetidine
N-[2-(3-methoxyphenyl)-1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-(3-aminopyrrolidine-1-carbonyl)-6-(2,5-dimethylfuran-3-yl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-{4-[7-chloro-3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)quinolin-2-yl]piperazin-1-yl}ethan-1-one
6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-9H-purin-2-amine
N-[(3-chloro-4,5-diethoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
(5-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}furan-2-yl)methanol
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]amine
6-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-1-yl)-9H-purine
3-(4-chlorophenyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
(3S,4R)-3-ethyl-4-methyl-1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-ol
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
6-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
{4-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}methanol
(2R,6R)-4-{[4-(2-hydroxyethoxy)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
8-[1-(4-fluorophenyl)piperidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
({6-[4-(2-methoxyethoxy)phenyl]pyridin-3-yl}methyl)dimethylamine
1-cyclopentyl-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-2-one
1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3-[2-(N-methylmethanesulfonamido)ethyl]urea