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1-(4-benzylpiperidin-1-yl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propan-1-one
N-cyclopropyl-1-[2-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}benzaldehyde
3-[4-(benzyloxy)piperidine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
1-cyclobutanecarbonyl-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3-methylpyridin-2-yl)formamido]acetic acid
N-cyclohexyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-propyl-1,2-oxazole-3-carboxamide
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
N-{3-[cyclopentyl(methyl)amino]propyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[6-chloro-2-(pyrimidin-5-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
2,6-dimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinoline-4-carboxamide
methyl 6-benzoyl-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-methyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
ethyl 1-(1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-4-carboxylate
3-(1H-indol-6-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-2-methoxypyridine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(3,4,5-trimethoxybenzoyl)piperidine
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-7,8-dimethylquinoline
3-(1-methylpiperidin-3-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
N-{1-[(4aS,7aR)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
N1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pentane-1,5-diamine
(3R,9R)-11-(4-fluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[1-(phenoxymethyl)cyclopropyl]methyl}piperidine-3-carboxamide
6-methyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1-(pyrrolidin-1-yl)ethan-1-one
1-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-methoxypropan-1-one
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{[1-(dimethylamino)cycloheptyl]methyl}-4-methylpyrimidin-2-amine
N-[(4,6-dimethylpyridin-2-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-(5-methoxy-2-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-(3,3-diphenylpiperidine-1-carbonyl)-1-methylpiperidin-4-ol
[(3R,4S)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}acetic acid
N-cycloheptyl-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-(1-propylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
3-{1-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
2-[4-(1-benzofuran-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-methyl-4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperazin-2-one
3-{[1-(2-methoxybenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[2-(dimethylamino)ethyl]-3-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)propanamide
2-{[4-(propan-2-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-methylfuran-2-carboxamide
4-({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
1-[2-(azepan-1-yl)-2-phenylethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-3-ylmethyl)piperidin-2-one
3-(4-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperazin-1-yl)-1-azabicyclo[2.2.2]octane