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1-(2-fluoro-5-methanesulfonamidophenyl)-3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]urea
4-[1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
2-methylpropyl 2-methyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
7,7-dimethyl-2-(pyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-[2-(piperidine-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-[2-(butan-2-yloxy)phenyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxolane-2-carboxamide
2-[4-({methyl[2-(pyridin-3-yl)ethyl]amino}methyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[(2R)-2-hydroxypropanoyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
5-(1-{5-[(2E)-pent-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
2-amino-6-[4-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]-3,4-dihydropyrimidin-4-one
[(3R,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2,3-dihydro-1H-inden-2-amine
N-methyl-5-{[methyl({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]methyl}pyrimidin-2-amine
(3R,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
2-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]-N-(2,3,4-trifluorophenyl)acetamide
1-{1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
methyl 2-[({2-[(2-chlorophenyl)methoxy]-7-fluoroquinolin-3-yl}methyl)amino]-4-(methylsulfanyl)butanoate
3-{[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-propylbenzamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
6-acetamido-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyridine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
2-[3-(2,3-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-azabicyclo[2.2.1]heptane
1-(cyclobutylmethyl)-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
(1-{1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
4-[4-(2,3-difluoro-4-pentylphenyl)-1H-pyrrole-2-carbonyl]morpholine
(3R,5S)-N-cyclopentyl-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3-carboxamide
2-phenyl-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}morpholine
5-ethyl-4-[3-(2-fluorophenoxy)azetidin-1-yl]pyrimidin-2-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(4-methoxyphenoxy)benzamide
1-(3-phenylpiperidin-1-yl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
(3R,4R)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-ethylpiperidine-3,4-diol
(5S)-5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
8-(2-hydroxy-3-methylbenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
{3-methyl-1-[3-({1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)benzoyl]piperidin-3-yl}methanol
3-(2-methylphenyl)-3-phenyl-1-[4-(pyrazin-2-yl)piperazin-1-yl]propan-1-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethyl-5,6-dihydro-1,4-dioxine-2-carboxamide
4-methyl-5-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
2-(dimethyl-1,2-oxazol-4-yl)-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}acetic acid
4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazine-2-carboxylic acid
2-cyclopropyl-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-amine
N-(cyclobutylmethyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(oxolan-2-ylmethyl)acetamide
N-[3-(4-fluoro-2-hydroxyphenyl)phenyl]acetamide
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxylate
3-[(3R,4S)-1-[(2,3-dichlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine