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4-(4-hydroxybenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
1-[(4-tert-butylphenyl)methyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[(2S)-3-methylbutan-2-yl]piperidin-4-amine
(1s,4s)-4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
N-(2-fluoro-4-methylphenyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]propanamide
1-[2-methoxy-5-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-(4-{[(2S)-2-benzyl-3-oxopiperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
4-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
N-ethyl-3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
2-[2-(3-acetamidopyrrolidin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2R,6S)-4-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-2,6-dimethylmorpholine
1'-(4-methylbenzoyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]quinolin-8-ol
(2S,4R)-1-(1-benzylpiperidin-4-yl)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
(3S,4S)-1-[(3-methylpyridin-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidin-4-yl)thiomorpholine
1-ethyl-N-[(2-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-methanesulfonyl-N-[3-(2-methoxyacetamido)phenyl]piperazine-1-carboxamide
2-{3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]morpholine-4-carbonyl}-3,4-dihydroquinazolin-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
(2S,3R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxybutanamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pentanamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(pyridin-4-yl)quinoline-4-carboxamide
2-(4-carbamoylpiperidin-1-yl)-2-(4-chloro-2,6-dimethoxyphenyl)acetic acid
N-cyclopropyl-2-(pyridin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
3-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}pyridine
5-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(2-benzylmorpholin-4-yl)-3-(2-fluorophenyl)propan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(2-methylphenyl)cyclopropyl]benzamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-7-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
6-ethyl-5-methyl-N4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-2,4-diamine
4-(2-chloro-6-methoxyphenyl)thiophene-2-carboxamide
2-benzyl-9-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)benzamide
4-[(4-methoxyphenyl)methyl]-1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,4-diazepan-5-one
9-(4-chloro-2-methylbenzoyl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(piperidin-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
(3R,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyridin-2-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
2-[2-(dimethylamino)ethyl]-9-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-cyclopropanecarbonyl-8-(6-methylpyridine-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3,5-dichloro-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-4-methylbenzamide