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3-acetamido-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)propanamide
1-(2-fluorophenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]cyclopropane-1-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(3S,4S)-4-cyclopropyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
ethyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(2-oxopyrrolidin-1-yl)benzamide
1-{[3-(2-methoxyethyl)-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,3-benzodiazole
4-(4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
4-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}benzoyl)morpholine
1,5-dimethyl-4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
5,7-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
methyl 1-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
3-{[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-1-ol
2-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(pyridin-2-yl)acetyl]piperidine-2-carboxamide
5-(oxolan-2-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
3-(5-{3-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]propyl}-1H-1,2,4-triazol-3-yl)pyridine
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[4-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(diethylamino)ethyl]-N-methyl-2-(4-propanoylphenoxy)acetamide
1-cyclopropanecarbonyl-4-[2-(4-fluorophenyl)azetidine-1-carbonyl]piperidine
4-hydroxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
2-{5-[1-(1,2-benzoxazol-3-yl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-cyclopentyl-3-methoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
2-(1-ethylpiperidin-4-yl)-1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
5-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-2-hydroxybenzoic acid
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(4-chlorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}butanamide
2-{[(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
5-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
2-[(1H-imidazol-2-ylmethyl)[(2-methylphenyl)methyl]amino]ethan-1-ol
1-[(3S,4R)-1-[3-(benzylsulfanyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methoxybenzene-1-sulfonamide
3-cyclohexyl-4-[(3-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{ethyl[2-(4-methylbenzenesulfonyl)ethyl]carbamoyl}benzoic acid
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)propanamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dipropylacetamide
9-methoxy-7-(4-methoxyphenyl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
[(3R,4S)-1-[(2,4-dimethylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[4-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-[4-(hydroxymethyl)phenyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(3aR,6aR)-2-(5-methyl-1,3,4-thiadiazol-2-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-(pyridin-3-ylmethyl)pyridin-2-amine