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7-(5-chloropyridine-2-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-methyl-1-(3-oxo-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propyl)-1,2-dihydropyridin-2-one
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-1-phenylethan-1-ol
(3R,4S)-4-cyclopropyl-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrrolidin-3-amine
2-ethyl-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-methoxy-1-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepan-1-yl)ethan-1-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyrazin-2-amine
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(2-methoxyethyl)acetamide
methyl 2-[(3-{4-[(2-methylpropyl)carbamoyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)sulfonyl]benzoate
(1S,5R)-6-[2-(2-ethoxyethoxy)benzoyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-[benzyl(methyl)amino]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
7-(5-chloropyridin-2-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-1-(3-chlorobenzoyl)-4-cyclobutyl-3-methylpiperidin-4-ol
1-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
2,2-dimethyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-cyclopropylacetamide
5-(1-{5-[2-methoxy-5-(propan-2-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
(5S,9aS,9bS)-5-[2-(dimethylamino)-1,3-thiazol-5-yl]-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-8-(trifluoromethyl)quinoline
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-(4-methoxyphenoxymethyl)piperidine-1-carboxamide
N-cyclohexyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aR)-2-(2-methoxyethyl)-5-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-ol
(2S,4S)-N-ethyl-4-[2-(methylsulfanyl)acetamido]-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-1-benzofuran-5-carboxamide
ethyl 3-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanoate
methyl[1-(pyridin-3-yl)ethyl](quinolin-2-ylmethyl)amine
2-amino-4-(4-hydroxy-3,5-dimethylphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
methyl 1-[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carbonyl]piperidine-2-carboxylate
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2,5-dimethylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-acetyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzene-1-sulfonamide
6-butyl-2-(4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
1,3-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(2,4-dichloro-6-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(1-methoxypropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopentyl-1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
(4aS,7aR)-1-{2-[(2-hydroxyethyl)(methyl)amino]acetyl}-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,7S)-N-[2-(dimethylamino)ethyl]-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
(4aS,8aS)-2-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
N-(2-hydroxyethyl)-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-indole-2-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-4-(pyridin-4-yl)pyrimidine