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6,7-dimethoxy-4-(piperidin-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-tert-butyl-4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
(1S,6R)-9-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
[(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
(1S,3R)-N-(3-fluorophenyl)-3-[2-(3-methoxyphenoxy)acetamido]cyclopentane-1-carboxamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
1-{[4-methoxy-3-(4-methoxy-3-methylphenoxy)phenyl]methyl}pyrrolidine
2-tert-butyl-4-hydroxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrimidine-5-carboxamide
3-{2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-(4-methanesulfonylpiperazine-1-carbonyl)-3,5-dimethyl-1H-indole
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
5-phenyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-2-(3-chloro-4-fluorophenyl)acetic acid
2,3-dimethyl-7-[3-(3-methyl-1H-1,2,4-triazol-5-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
7-(2-methylphenyl)-4-(6-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(2-{1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
2-(4-{[2-(difluoromethoxy)phenyl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
1-[(3-methylphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
2-{4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
2-(3-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(quinolin-5-ylmethyl)propanamide
N-[3-(benzylsulfanyl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-(tert-butylamino)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
3-{1-[6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]-N-methylformamido}propanamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1-methylpiperidin-3-yl)methyl]pyridin-2-amine
2,7,8-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]quinoline
1-{4-[3-({[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
1-(1-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}ethyl)-4-methylpiperazine
1-methyl-6-(pyridin-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-amino-1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(1H-1,2,3-triazol-4-ylmethyl)pyrrolidin-3-yl]butane-1-sulfonamide
5-cyclopropanecarbonyl-1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-(oxolan-3-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-[4-(2-methylphenyl)piperazin-1-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-cyclopropyl-6-[4-(1-methoxyethyl)phenyl]pyrimidine
1-methyl-N-[2-(methylsulfanyl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(4-acetylmorpholin-2-yl)methyl]-1-[3-(2-ethoxyethoxy)phenyl]urea
3-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)phenol
3-[2-(oxan-2-yl)ethyl]-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-chloro-6-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]pyridine-2-carboxylic acid
8-[(2,6-difluorophenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1H-imidazole-5-carbonyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3R,4R)-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide