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(1S,5R)-3-(5-chloro-3-fluoropyridin-2-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-(cyclopropylmethyl)-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-cyclobutanecarbonyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(5-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetate
2-{3-oxo-9-[2-(phenylsulfanyl)acetyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(1S,5R)-6-[4-(propan-2-yloxy)benzoyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
9-(2-aminopyrimidin-4-yl)-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[(2-aminopyrimidin-5-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
1,7-dimethyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-indole-2-carboxamide
N-cycloheptyl-N-methyl-3-[methyl(1-methylpyrrolidin-3-yl)amino]propanamide
3-{5-[(4-cyanophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopentylpropanamide
4-[(dipropylamino)methyl]-N-(pyrrolidin-3-yl)benzamide
1-{[4-(cyclopentyloxy)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidin-4-ol
3-(3-{2-[2-(difluoromethoxy)phenyl]-1H-imidazol-1-yl}propyl)pyridine
2-[3-(methylsulfanyl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-propoxypropanamide
(3S,4R)-4-(4-fluorophenyl)-1-(quinolin-4-ylmethyl)pyrrolidine-3-carboxylic acid
3-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(pyridin-4-yl)ethyl]benzamide
3-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
5-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
4,6-dimethoxy-2-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidine
4-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-N-methylbenzene-1-sulfonamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methylpyridine
4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
4-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-N-methylpyridin-2-amine
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(morpholin-3-yl)acetamide
N-methyl-3-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)pyridin-2-amine
4-({2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(azocan-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-benzyl-4-(3-hydroxypropyl)-1-(4-methylphenyl)piperazin-2-one
3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]phenol
ethyl 4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
N-cyclopropyl-3-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}sulfonyl)benzamide
3-[3-(3-methylphenoxy)azetidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
9-ethyl-4-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(1-methoxypropan-2-yl)-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine-4-carboxamide