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(3R,9aR)-3-(hydroxymethyl)-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(2S)-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-N-methyl-1-[(E)-2-phenylethenesulfonyl]pyrrolidine-2-carboxamide
5-(4-oxo-4H-chromen-3-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
4-({[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]amino}methyl)-1-cyclopropylpyrrolidin-2-one
8-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-[(3,5-dimethylphenyl)methyl]-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-2-one
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
1-[(4-fluorophenyl)methyl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N3-cyclohexyl-1-cyclopropyl-N5-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{4-[2-(thiophen-3-yl)acetyl]morpholin-3-yl}acetamide
2-(1-{[4-(methylsulfamoyl)phenyl]methyl}piperidin-2-yl)acetic acid
1-(2-methoxyethyl)-4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-(adamantan-1-yl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)acetamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
4-methyl-N-[3-(methylsulfanyl)propyl]-3-phenyl-1H-pyrazole-5-carboxamide
1-ethyl-4-{[(5-ethylpyrimidin-2-yl)(methyl)amino]methyl}pyrrolidin-2-one
8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,8-diazaspiro[4.5]decan-3-one
5,7-dimethyl-N-[3-(pyridin-2-yl)propyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
(2S,4R)-1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(dimethylamino)pyrrolidine-2-carboxylic acid
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-amine
(1S,5R)-3-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
4-{[5-(1-ethylpiperidin-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,5-dimethylpyrazine-2-carboxamide
N-cyclopropyl-1-ethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-3-carboxamide
6-fluoro-4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
6-fluoro-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
4-(2-methoxyphenyl)-2-{4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyrimidine
6-ethyl-2-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}quinoline-4-carboxamide
3,5-dichloro-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,4-dimethylbenzamide
N-[2-(dimethylamino)ethyl]-5-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-ethyl-5-(1-{[4-(pyridin-2-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(4-methyl-1,3-thiazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(4-fluorophenyl)cyclopropane-1-carboxamide
N-(butan-2-yl)-N-(pyridin-4-ylmethyl)-1,2,3-thiadiazole-4-carboxamide
(3aR,6aR)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(3-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-[6-amino-5-cyano-4-(1-ethyl-1H-indol-6-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
4-{4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}phenol
2-(morpholin-4-yl)-8-(2,4,5-trifluorophenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
(2S)-3-phenyl-2-[2-(4-propanamidophenoxy)acetamido]propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-1-methylpiperidine-3-carboxamide
(3aR,6aS)-5-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(2,5-dimethylfuran-3-yl)methyl]piperazin-1-yl}phenol