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3-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
(5-{[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-(methylsulfanyl)ethan-1-one
8-[3-methyl-4-(morpholin-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
4-(2H-1,3-benzodioxol-5-yl)-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,9aR)-1-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(dimethylamino)ethyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}benzamide
N-[(2,3-dimethoxyphenyl)methyl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2-methylphenyl)methyl]-3-(1,2-oxazinan-2-yl)-N-(oxolan-2-ylmethyl)propanamide
5-(1,5-dimethyl-1H-indazol-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-9-oxa-2-azaspiro[5.5]undecane
2-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-fluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzene-1,2-diol
1-methyl-4-phenyl-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
3-({[1-(2-chloro-6-fluoro-3-methylbenzoyl)piperidin-3-yl]oxy}methyl)pyridine
N-[3-(cyclohexylsulfanyl)propyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
(2S,4R)-N,N-diethyl-4-(furan-3-amido)-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(furan-2-carbonyl)-1,4-diazepane
1-[2-(dimethylamino)ethyl]-4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)pyrrolidin-2-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(2-phenylethyl)pyrrolidin-2-one
(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]piperidin-3-yl)methanol
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
1-[3-phenyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
5-({methyl[(3-{2-[4-(4-methylbenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
2-(2-{1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(2R,3R,6R)-3-(4-methylphenyl)-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]acetamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
6-({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carbonitrile
1-[2-(dimethylamino)ethyl]-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(hydroxymethyl)azepan-4-ol
[3-(3-methoxypropyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]methanol
methyl 3-(2-methoxyacetamido)-5-{[(4-methylphenyl)formamido]methyl}benzoate
N-[2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-N-propylaniline
2-(2-methyl-5-propylpyrimidin-4-yl)-1,2,3,4-tetrahydroisoquinolin-4-ol
(5S,9aS,9bS)-5-[4-ethoxy-3-(hydroxymethyl)phenyl]-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-(thiophen-2-ylmethyl)-6-[4-(thiophene-2-carbonyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}propanamide
1-[4-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-oxoethoxy)phenyl]propan-1-one
2-{4-[(4-phenylphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
4-(1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-methylpropan-2-yl)morpholine
N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-1,3-benzodiazole-2-carboxamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-indazole-3-carboxamide