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N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
2-{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
ethyl 2-{[3-(3-methylthiophene-2-carbonyl)piperidine-1-carbonyl]amino}acetate
(2S,4S)-4-amino-N-ethyl-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
2,6-difluoro-N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}benzamide
1-[3-(3-methylphenyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(3S,4S)-1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]-4-(morpholin-4-yl)butanamide
N-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]morpholine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2,4,5-trimethylphenyl)methyl]piperidine
2-methyl-N-[(1-methylpiperidin-3-yl)methyl]-4-phenyl-1,3-thiazole-5-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-ethoxyethan-1-one
1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3-phenylpyrrolidin-3-ol
8-(2-aminopyrimidin-4-yl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
6-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
11-{[(4-fluorophenyl)methyl]amino}-4-[2-(3-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(4aS,7aR)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-cyclopentyl-N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]pyrimidin-2-amine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
(1S,4S)-2-[2-(4-chloro-2-methylphenoxy)ethyl]-2-azabicyclo[2.2.1]heptane
1-(5-chloropyridin-2-yl)-4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperazine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methylacetamide
(3R,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-ethyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2-chlorophenyl)-3-{1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N4-methyl-6-(morpholin-4-yl)-N4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-2,4-diamine
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
N-[(3R,4S)-1-[2-(azepan-1-yl)acetyl]-4-phenylpyrrolidin-3-yl]acetamide
(2R,6R)-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-4-carboxamide
3-[(1-methylpiperidin-4-yl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
2-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-methylpyridine
1-[4-(2-methylpropyl)-1,4-diazepan-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-(furan-3-ylmethyl)-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
N'-(3-chloro-2-methylphenyl)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]propanediamide
1,3-dimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methoxy-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
1-(2-chloropyridin-3-yl)-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}urea
3-(3-methoxyphenyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
3-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-(3,4,5-trimethoxyphenyl)urea
4,5,6-trimethyl-2-oxo-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1,2-dihydropyridine-3-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]propan-1-one
3-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-N-(3-methylphenyl)propanamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
(3R,4S)-4-[ethyl({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)amino]oxolan-3-ol