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3-({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-1,1,1-trifluoropropan-2-ol
2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
N,N-dimethyl-2-[({[(1S)-1-phenylpropyl]carbamoyl}amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-{4-[4-(3-fluoropyridin-4-yl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
dimethyl(3-{2-[1-(pyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(quinolin-4-ylmethyl)amine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-methoxy-5-{1-[1-(4-methylpyridin-2-yl)propyl]-1H-1,2,3-triazol-4-yl}pyridine
(2S)-2-amino-3-hydroxy-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(cyclobutylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
diethyl({3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(3aS,6aS)-2-methyl-5-[(3-methylpyrazin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-{[4-(2-fluorophenoxy)phenyl]carbamoyl}piperidin-1-yl)propanoic acid
(3S,7S)-5-(pyridine-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-[cyclopropyl(1,3-thiazol-5-ylmethyl)amino]-N-[1-(4-methylphenyl)ethyl]acetamide
N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-{[2-(difluoromethoxy)phenyl]methyl}-N-phenylpiperidin-3-amine
(4aR,7aS)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(furan-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
N,N-dimethyl-4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(methylsulfanyl)acetamide
3-{3-[3-(5-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
3-[({[1-(4-methoxyphenyl)cyclopentyl]methyl}amino)methyl]pyrrolidin-3-ol
2-(propan-2-yl)-5-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,3-benzoxazole
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
1-(2-methylpyridin-4-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{3-[(pyridin-3-yl)amino]propyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(3ar,6ar)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[4-chloro-3-({[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
1-[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
4-{[2-(2-fluorophenyl)ethyl]amino}-N,N,5-trimethylthieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(diphenylmethyl)piperazin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
[(3R,4R)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{[2-(1-ethylpiperidin-4-yl)acetamido]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methylpentyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-hydroxyphenyl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]-1H-pyrazole-5-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(4-{2,8-diazaspiro[4.5]decane-3-carbonyl}piperazin-1-yl)pyridine-3-carboxamide
5-phenyl-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
({4-ethyl-5-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(3-methylthiophen-2-yl)methyl]amino}pyrrolidin-2-one
N-[2-(dimethylsulfamoyl)ethyl]-3-methyl-1-benzothiophene-2-carboxamide
6-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
2-amino-4-(4-hydroxyphenyl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-(oxolan-2-ylmethyl)-2-{4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}acetamide
4-(1-hydroxy-3-methylbutan-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one