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1-(3-phenylpropyl)-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
2-ethyl-4-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-5-carboxamide
2-[4-(6,8-dimethylquinolin-4-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
5-{[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]methyl}-2-methoxybenzoic acid
1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
(3S,4S)-4-cyclopropyl-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)pyrrolidine-3-carboxylic acid
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(thiophen-2-ylmethyl)piperazine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-cyclopropyl-3-methyl-1H-pyrazole-4-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-indol-1-yl)ethan-1-one
3-methyl-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-phenylpiperazin-2-one
1-(cyclopropylmethyl)-N-ethyl-5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-4-methylpentane-1,2-dione
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-9H-purine
5-[({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}amino)methyl]-1,2,4-oxadiazole-3-carboxamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4-phenylbutane-1,2-dione
methyl 4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}thiophene-2-carboxylate
2-({4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperazin-1-yl}methyl)benzonitrile
1-[4-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(4-methylphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-cyclopropanecarbonyl-2-(2-methylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(5-methylthiophene-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
5-ethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(4aS,8aR)-6-[4-(1H-imidazol-1-yl)butanoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-[(5-oxopyrrolidin-2-yl)methyl]-5-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
3-(1H-imidazol-2-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine
2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
1-(4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenyl)ethan-1-one
1,7-dimethyl-2-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1H-indole
4-[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-ol
3-{[6-oxo-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(furan-3-ylmethyl)-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-ethyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidine-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-[(2-fluorophenyl)formamido]propanamide
ethyl 2-(N-methyl-1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazol-3-yl}formamido)acetate
(3S)-1,3-dimethyl-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
1-(cyclopropylmethyl)-5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
5-{[4-(methylsulfanyl)phenyl]methyl}-5-{3-oxo-3-[3-(3-phenylpropanoyl)piperidin-1-yl]propyl}pyrrolidin-2-one
4-[(2-chlorophenyl)methyl]-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
(2R,3R)-3-(dimethylamino)-1'-{thieno[2,3-d]pyrimidin-4-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-methanesulfonyl-4-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazine
2-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-fluorobenzene-1-sulfonamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide