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(3S)-4-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,3-dimethylpiperazin-2-one
1-(cyclohexylmethyl)-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-{[3-(1-phenylcyclobutyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
2-{[2-(adamantan-1-yl)-4-hydroxypyrimidin-5-yl]formamido}-N-(propan-2-yl)acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(morpholin-4-yl)butanamide
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
2-(3-cyclopropyl-1-ethyl-1H-1,2,4-triazol-5-yl)-3,4,7-trimethyl-1H-indole
2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-N-(2-methoxy-5-methylphenyl)acetamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(3-methoxyphenyl)methyl]piperidine
1-(2,3-dimethylphenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
1-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-3-methoxy-1,2-dihydropyridin-2-one
2-{4-[(3,5-difluorophenyl)methyl]piperazine-1-carbonyl}-1-methylazepane
4-fluoro-2-[({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)methyl]phenol
4-[4-(3-cyanopyridin-2-yl)piperazin-1-yl]-N-cyclopentyl-4-oxobutanamide
4-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1R,2S)-2-phenylcyclopropyl]pyrimidine-5-carboxamide
2-cyclopentyl-8-(trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
8-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1λ6-thiane-1,1-dione
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidin-3-yl)benzamide
1-(4-methoxyphenyl)-5-methyl-4-(pyrrolidine-1-sulfonyl)piperazin-2-one
4-(4-{1-[(3-methylphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)butanamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(piperazin-1-ylmethyl)piperidin-2-one
9-[2-(4-ethoxyphenyl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(4aS,8aR)-6-(4,6-dimethylpyrimidin-2-yl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(2-chloropyridin-3-yl)methyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
(1R,3S)-3-methoxy-7-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-7-azaspiro[3.5]nonan-1-ol
N-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
4-(cyclopropylmethyl)-1-[2-(4-methylphenyl)quinoline-4-carbonyl]-1,4-diazepan-5-one
N-[(1R,3R)-3-aminocyclopentyl]-2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
N-methyl-3-{1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperidin-3-yl}-N-(1-methylpiperidin-4-yl)propanamide
(4-{[methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})amino]methyl}oxan-4-yl)methanol
2-(adamantan-1-yl)-4-hydroxy-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidine-5-carboxamide
1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-2-yl)acetamide
1-ethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-cyclopropyl-N-(4-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)propanamide
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[(2S,4R,6R)-2-(2-amino-1,3-thiazol-5-yl)-6-cyclohexyloxan-4-yl]acetamide
(3S,5S)-5-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-1-methylpyrrolidin-3-amine
3-[2-(2-methyl-1H-indol-3-yl)ethyl]-3,4-dihydropteridin-4-one
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-{8-[(4-methoxyphenyl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-(3-phenylpropyl)-8-(pyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-benzyl-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1,3-benzoxazole-5-carboxamide
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one