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2-(3-hydroxypropyl)-9-[2-(methylamino)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-methoxypyridin-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-butyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
N,N-diethyl-3-[methyl(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-methylcyclopropyl)acetamide
(3aR,7aS)-2-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-(piperidin-1-ylmethyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-ol
2-methyl-4-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-6-propylpyrimidine
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(3-methylpyridin-2-yl)piperazine
1-(1-benzothiophen-5-ylmethyl)-4-methylpiperazine
N-(2,6-difluorophenyl)-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
methyl 4-(5-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
dimethyl(2-{2-[1-(thiophene-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-methyl-3-(piperidin-3-yl)-N-(quinolin-4-ylmethyl)benzamide
N-[4-(oxolan-2-yl)butyl]-6-(propan-2-yl)pyrimidin-4-amine
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[(4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)methyl]-5-methyl-1H-1,2,3,4-tetrazole
7-(cyclobutylmethyl)-2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-[(5-methylthiophen-2-yl)methyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
4-(4-ethoxy-3-methylphenyl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}butanamide
(4S)-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3,3,4-trimethylpiperidin-4-ol
1-[2-(dimethylamino)-4-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[4-(3-methylfuran-2-carbonyl)morpholin-3-yl]-N-[2-(pyridin-3-yl)ethyl]acetamide
2-methyl-7-(oxolan-3-ylmethyl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-3-(pyridin-2-ylmethyl)-6-[4-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-({5-[1-(furan-3-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
(1S,9R)-11-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-{1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-3-(2,5-dioxoimidazolidin-4-yl)propanamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
8-(4-ethyl-5-methylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-{1-[(methylcarbamoyl)methyl]-1H-pyrazol-4-yl}-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-methyl-4-{[methyl(1-methylpyrrolidin-3-yl)carbamoyl]amino}benzamide
5-[2-(2-ethoxyethoxy)phenyl]-3-phenyl-1H-1,2,4-triazole
N-{[1-(4-phenylbenzenesulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
N-ethyl-N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-4-yl)benzamide
1-[(5-chlorothiophen-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-6-(methoxymethyl)pyridine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]propanamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
dimethyl[(5-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}thiophen-3-yl)methyl]amine