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1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-hydroxyethan-1-one
5-cyclopropanecarbonyl-1'-[(3-fluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{butyl[2-(cyclohex-1-en-1-yl)ethyl]amino}butan-1-ol
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(azepan-1-yl)-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(3aS,6aS)-2-methyl-5-{[4-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-phenyl-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
2-{[(2-chlorophenyl)methyl](methyl)amino}-2-(2,5-dimethoxyphenyl)acetic acid
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-methylbenzamide
(4aR,8aR)-4-[3-(1H-1,2,4-triazol-3-yl)benzoyl]-octahydro-2H-1,4-benzoxazine
3-[2-(2-methylphenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
7-(3-chlorophenyl)-4-(1-hydroxycyclopentanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(3R,4S)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2,4-dimethyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
benzyl(cyclopropylmethyl){[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
7-(2-ethylphenyl)-1,2-dihydroisoquinolin-1-one
3-(6-methoxyquinolin-8-yl)-1-(oxan-4-yl)urea
N-{1-[1-(4-chloro-3-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
4-methyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,3-thiadiazole
1-methyl-9-(2-propylpyridine-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}morpholine
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
4-({5-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)phenol
3-cyclopropyl-5-(methoxymethyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N4-ethyl-N2-methyl-N2-[2-(morpholin-4-yl)propyl]pyrimidine-2,4-diamine
2-({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
(3R,4S)-N,N-dimethyl-4-propyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)(propan-2-yl)amine
2-ethyl-4-methyl-5-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,3-thiazole
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[4-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(pyridin-4-yl)ethyl]acetamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-(phenylamino)pyrimidine-5-carboxamide
1-[1'-(2-cyclohexylacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-6-methoxyphenol
ethyl 4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
2-(3-methoxypropyl)-8-(2-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[4-({1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxane-4-carboxamide
N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-4,4-difluoropiperidine-1-carboxamide
3-(4-chlorophenyl)-4-{[1-(propan-2-yl)piperidin-4-yl]formamido}butanoic acid
3-{5-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
2-[2-(2-methylpropoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine