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1-(1-propylpiperidin-4-yl)piperidine-3-carbonitrile
N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}propane-1-sulfonamide
{3-cyclopentanecarbonyl-9-[(2-methyl-1H-imidazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(1S,5R)-3-(3-chloro-2-methylbenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethylamino)butan-1-one
1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[5-(2-cyclopropylquinolin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]butan-2-ol
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(4-fluorophenoxy)piperidine
5-acetyl-N-{[2-(benzyloxy)phenyl]methyl}thiophene-3-carboxamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline
4-{1H-imidazo[4,5-b]pyridin-2-yl}-1-methyl-3-(4-phenoxyphenyl)-1H-pyrazole
2-phenoxy-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}butan-1-one
1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-4-(thian-4-yl)piperazine
1-(2-methoxyethyl)-N-[2-(3-methylthiophen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1H-imidazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aS)-2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
2-(2,3-dihydro-1H-indol-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-oxoacetamide
[(3R,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3S,4S)-N-(4-chloro-2,6-dimethylphenyl)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
6-methyl-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydroquinoline-4-carboxamide
5-(phenoxymethyl)-N-(1-propylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
(2R)-2-amino-2-cyclohexyl-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
[5-(8-methoxyquinolin-5-yl)-1H-1,3-benzodiazol-2-yl]methanol
(2S,4S)-4-amino-N,N-diethyl-1-(2-fluoro-4-methylbenzenesulfonyl)pyrrolidine-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
[(2S,4R)-4-(dimethylamino)-1-[1-(piperidin-1-yl)cyclohexanecarbonyl]pyrrolidin-2-yl]methanol
2-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,3-benzodiazole
4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]pyridine-3-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-(4-methoxy-3-methylphenyl)-6-methyl-9H-purine
1-(3-fluorophenyl)-3-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-(3-ethylphenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
8-[3-(methylsulfanyl)propanoyl]-2-(phenoxymethyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-4-(piperidin-3-yl)benzamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propan-1-one
2-(5-methyl-1H-pyrazol-1-yl)-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[3-(methylsulfanyl)propyl]pyrimidine-5-carboxamide
3-chloro-N-(2-methoxyethyl)-4-({1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazol-2-yl]-2-(pyridin-2-yl)pyrimidine
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-yl)pyridin-2-amine