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N-benzyl-N-methyl-3-[(4-methyl-1,4-diazepan-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
4-phenyl-1-(thian-4-yl)azepane
5-[(3-fluoro-4-methylphenyl)methyl]-3-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-(4-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(1H-indole-6-carbonyl)-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-fluorophenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-one
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(3-methoxyphenyl)-2,2-dimethylpiperazine
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3,3-dimethylbutan-1-one
1-(3-methylbutyl)-8-(pyridin-3-ylmethyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N'-(3,5-dimethylphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanediamide
2-(4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
(3S,7S)-5-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(3-methoxypyridin-2-yl)-N,N-bis(propan-2-yl)benzamide
3-cyclohexyl-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazole
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
3-(3-fluorophenyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
N-[3-(1H-imidazol-1-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[3-methyl-4-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
6-[({2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N2,N2-dimethyl-1,3,5-triazine-2,4-diamine
2-(2-phenylethyl)-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}morpholine
2-{[1-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N,N-dimethylethane-1-sulfonamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(1-propylpiperidin-4-yl)pyrimidin-2-amine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
2-(2,5-dimethylphenoxy)-N-ethyl-N-(4-hydroxybutyl)propanamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-[3-(4-methoxyphenyl)propyl]-6-(1H-pyrazol-3-yl)pyridine-3-carboxamide
N-methyl-3-(2-phenoxyethyl)benzamide
(3R,4R)-3-cyclobutyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-methylpyrrolidin-3-ol
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
{5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]furan-2-yl}methanol
2-[3-(5-methylfuran-2-yl)-5-(3-phenyl-1,2-oxazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-(1,4-dioxan-2-ylmethyl)-N-methyl-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]furan-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)benzamide
2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carboxamide
2-amino-4-ethyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1,3-thiazole-5-carboxamide
6-methyl-5-[5-(5-methyl-4-phenylthiophen-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(furan-2-ylmethyl)-3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-(2,6-dimethylphenoxy)-1-(quinoxalin-2-ylmethyl)piperidine-4-carboxylic acid
1-(1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(dimethyl-1,3-oxazole-5-carbonyl)piperidine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
4-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
ethyl 2-({methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)-1H-imidazole-5-carboxylate
3-(4-benzyl-1H-pyrazol-5-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
3-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
1-[(4aR,8aR)-4a-hydroxy-7-[(4-phenoxyphenyl)methyl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one