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N-[2-(2-fluorophenyl)-1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
N-(furan-2-ylmethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(prop-2-yn-1-yl)-1H-pyrazole-3-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
5-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-ethyl-3-methyl-1H-pyrazole
2-{1-azabicyclo[3.2.1]octan-5-yloxy}-5,8-dimethoxy-4-methylquinoline
N-{2-methoxy-4-[2-(5-oxopyrrolidin-2-yl)acetamido]phenyl}-2,2-dimethylpropanamide
(2S,4R)-4-amino-N,N-diethyl-1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidine-2-carboxamide
2-(propan-2-yl)-5-(1-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1H-imidazol-2-yl)pyrimidine
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
9-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(3-methoxybenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
N-cyclopentyl-6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
6-[methyl(pyrimidin-4-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(3R,4S)-1-[(4-fluorophenyl)methanesulfonyl]-4-phenylpyrrolidin-3-amine
1-(1-cyclopentylpiperidine-3-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-{[4-(4-methoxyphenyl)-5-(oxan-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[(2R,3R,6R)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
3-(cyclopropylmethyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine-3-carboxylic acid
1-[3-(2-ethylphenoxy)azetidin-1-yl]-4,4,4-trifluorobutan-1-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(thiolan-3-yl)-1H-imidazole
3-butyl-4-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-methylpiperazin-2-one
2-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-tert-butyl-N-[(2-fluorophenyl)methyl]-4-hydroxy-N-(2-methoxyethyl)pyrimidine-5-carboxamide
(2S)-N-ethyl-1-[4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
1-[2-(diethylamino)acetyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
2-ethyl-N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]pyrimidine-5-carboxamide
2-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
N-{2-methyl-5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}cyclobutanecarboxamide
8-(4-ethyl-5-methylthiophene-3-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 6-[(2-hydroxyphenyl)methyl]-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[5-(1-cyclobutanecarbonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
5-butyl-1-(4-chlorophenyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
4-[1-(2H-1,3-benzodioxol-4-ylmethyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
7-ethyl-1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-methyl-5H,6H,7H,8H-imidazo[1,5-a]pyrazin-8-one
1-(cyclohexylmethyl)-N3-cyclopropyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(5-acetylthiophen-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
{4-[3-(3-fluorophenyl)benzoyl]-1,4-oxazepan-6-yl}methanol
2-methyl-4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]quinoline
2-hydroxy-4-(methylsulfanyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(3S,4S)-1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-propylpyrrolidine-3-carboxylic acid
N-[3-(3-chlorophenyl)phenyl]-1-(5-methylthiophene-2-carbonyl)piperidine-4-carboxamide
[(2-fluorophenyl)methyl](2-methoxyethyl)[(6-methoxypyridin-3-yl)methyl]amine