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(1-benzothiophen-2-ylmethyl)({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
8-(4-methyl-1H-pyrrole-2-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methyl-4-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-2-(thiophen-2-yl)-1,3-oxazole
N-cyclohexyl-3-{[1-(1H-pyrazol-1-yl)propan-2-yl]amino}propanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-4-yl)propanamide
4-methoxy-6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
(4aR,7aS)-1-(pyridin-3-ylmethyl)-4-(thiophene-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-4-hydroxy-N-[3-(1H-indol-1-yl)propyl]pyrimidine-5-carboxamide
N,N,8-trimethyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-(2-hydroxyethyl)-N-methyl-6-oxopiperidine-3-carboxamide
3-(2-methoxyethyl)-5-(3-methyl-5-propyl-1-benzofuran-2-yl)-1,2,4-oxadiazole
ethyl 2-{1-[5-(cyclooctylcarbamoyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridin-3-yl]-N-methylformamido}acetate
3-(2,6-dimethoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-(4-methyl-6-{4-[(oxolan-3-yl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1-benzoxepine-4-carboxamide
(2S,4S)-4-amino-1-{2-[3,5-bis(trifluoromethyl)phenyl]acetyl}-N-methylpyrrolidine-2-carboxamide
(3S,4S)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidine-3,4-diol
2-[4-(4-methyl-2-phenylpiperazine-1-carbonyl)piperidin-1-yl]acetamide
2-[benzyl(methyl)amino]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
6-(2-chlorophenyl)-N-(4-hydroxybutyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(2,4-dimethoxybenzoyl)-3,4-dihydro-2H-1,4-benzoxazine
N'-(3-chloro-2-methylphenyl)-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]propanediamide
3-(furan-2-yl)-2-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}propan-1-ol
1-methyl-4-{[5-(oxan-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
5-(dimethylamino)-2-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-5-(methoxymethyl)furan-2-carboxamide
1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-propoxyethan-1-one
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-diazepan-5-one
1-(cyclohexylmethyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
3-(azepane-1-carbonyl)-1-methyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(dimethylamino)-1-phenylpropyl]-5-methyl-1,3-oxazole-4-carboxamide
6-(3,5-dichloro-4-methylbenzoyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(1,3-benzothiazol-2-ylmethyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-(3-fluorophenoxy)-1-(3-methylfuran-2-carbonyl)piperidine-4-carboxylic acid
1-(2-fluorophenyl)-4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)piperidin-4-ol
(2S,4R)-4-[(adamantan-2-yl)amino]-N-ethyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
3-cyclopropyl-N-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,2,5-oxadiazole-3-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(2-methoxynaphthalen-1-yl)methyl]acetamide
(4aS,7aR)-1-[(5-ethylpyridin-2-yl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}-N-methylacetamide
N-[4-(4-{[2-(methylsulfanyl)ethyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
2-ethyl-N-[2-(ethylsulfanyl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
3,6,7-trimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
(2R,3S,6R)-5-(1-benzofuran-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-(morpholine-4-carbonyl)-1,4-diazepan-6-ol
4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
4-ethyl-1-methyl-3-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one