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2-methyl-5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-3,4-dihydropyrimidin-4-one
6-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3-methylquinoxaline
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
(9aS)-N-[3-(2-methoxyacetamido)phenyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
8-(2,3,4-trimethoxybenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-(3,4-dichlorophenyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)morpholine
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-phenyl-1,2-oxazole
(1R,5R)-N-[2-(2-fluorophenyl)ethyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(morpholin-4-yl)-3-[1-(thian-4-yl)piperidin-4-yl]propan-1-one
4-[2-(4-methoxyphenyl)ethyl]-11-[4-(propan-2-yl)piperazin-1-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
9-(2-hydroxyethyl)-1-methyl-4-(2-phenylacetyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5,6-dimethyl-1-(pyridin-4-yl)-1H-1,3-benzodiazole
N,5-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-benzofuran-2-carboxamide
(1S,5R)-6-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[(2,6-dichloro-3-hydroxyphenyl)methyl](methyl)amino}methyl)-1-methylpyrrolidin-2-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-[1-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-({4-methyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-(2-benzylmorpholine-4-carbonyl)-4-fluorobenzene-1-sulfonamide
(5-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(pyridin-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)urea
2-[4-({cyclohexyl[2-(ethylsulfanyl)ethyl]amino}methyl)-3,5-dimethyl-1H-pyrazol-1-yl]ethan-1-ol
1-{3-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-N-[2-(morpholin-4-yl)ethyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3-propylpiperidin-3-yl)methanol
N-(1-cycloheptylpiperidin-3-yl)-2-methylbenzamide
3-(4-methylphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
7-cyclohexyl-2-(2-methoxypyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-2-methoxyacetamide
N-methyl-N-(pyridin-3-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
6-(3-oxopiperazin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-methanesulfonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[2-(ethylsulfanyl)pyrimidin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)prop-2-yn-1-yl}morpholine
(2S,4R)-4-amino-1-(3,4-diethoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
7-(cyclobutylmethyl)-2-(quinoxaline-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-methoxy-2-(6-methoxy-2H-1,3-benzodioxol-5-yl)quinoline
4-(2-phenylethyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-(1-methyl-1H-pyrazol-3-yl)-4-(prop-2-en-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(4-fluorophenyl)ethyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}pyridin-2-amine
2-(3-hydroxypyridine-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
8-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one