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1-(2-chlorophenyl)-4-[2-(1H-indol-1-yl)acetyl]-5-methylpiperazin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-3-acetamido-N-methylbenzamide
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
1-[6-(6-methoxy-1H-indol-2-yl)pyridin-2-yl]ethan-1-ol
3-(2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butanamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N2,6-dimethylpyrimidine-2,4-diamine
(3R,4S)-1-(1-methyl-1H-imidazole-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[3-(methylsulfanyl)propyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-chloropyridin-3-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(4aS,8aR)-6-[3-(benzyloxy)propyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-{1-[3-(carbamoylmethyl)-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl]butyl}acetamide
2,4-dimethyl-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide
1-[(4-chlorophenyl)methyl]-5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-2-one
2-methoxy-N-(1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carboxamide
5-methyl-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-phenylpiperidin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-[3-(1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
(4aS,7aR)-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-phenylpiperazin-1-yl)-5-(thiophen-2-ylmethyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-methyl-N-[(1-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
[(3R,4R)-1-(2,3-dichlorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[(3R,4S)-1-(1-methyl-1H-indole-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
9-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-hydroxybutan-2-yl)-2-(methylsulfanyl)-N-(thiophen-2-ylmethyl)acetamide
[(3R,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-benzyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-methyl-4-oxo-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
N,N-bis(1,3-oxazol-4-ylmethyl)-5-phenyl-1H-pyrazole-3-carboxamide
8-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1H-indole-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-cyclobutanecarbonyl-N-[2-(3-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(oxan-4-yl)piperazine
methyl 5-[(1-phenyl-1H-pyrazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-({1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)-2-(furan-2-yl)-2-oxoacetamide
5-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)thiophene-2-sulfonamide
2-{2-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol