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2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophene-3-sulfonamide
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-(5-methoxyfuran-2-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-[2-(pyrrolidin-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
[(8-chloroquinolin-2-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
9-(4,6-dimethylpyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-5-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
4-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-2-(propan-2-yloxy)propanamide
(2S)-2-amino-3-cyclohexyl-N-(4H-1,2,4-triazol-4-yl)propanamide
6-(5-chloro-2-methoxyphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-{1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-2-yl}benzoic acid
2-ethoxy-3-{[4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(2-ethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2,6-dimethyl-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}quinoline
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(4-methoxybenzoyl)piperazine
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(2-fluorophenyl)-4-[(2-methylpyridin-3-yl)methyl]piperazine
6-fluoro-2-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
1-benzyl-4-[4-(4-chlorophenyl)butanoyl]piperazin-2-one
3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-methyl-1,3-oxazole
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-1,3-thiazole-5-carboxamide
1-{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
2-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
(1S,5R)-3-[(2-chloro-5-fluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-phenylpiperidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-cyclooctyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(2S)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
9-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4R)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-{9-[2-(4-methylphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
2-benzyl-9-(9H-purin-6-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-5-[2-(phenylformamido)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2R,3R,6R)-5-[(3-ethyl-1H-pyrazol-5-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aR)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(morpholin-4-yl)-1-(4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)ethan-1-ol
2-(dimethylamino)-N-{2-[ethyl(methyl)amino]-2-methylpropyl}-2-(2-methylphenyl)acetamide
3-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
4-[1-(2-phenyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]pyridine
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-[2-(azepan-1-yl)-2-phenylethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-chloro-5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(2-methoxyphenoxy)-1-(oxolan-3-ylmethyl)azetidine