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5-(2-hydroxy-5-methoxyphenyl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-(2,4-dimethoxyphenyl)-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
1-(4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
N-[2-(ethylsulfanyl)ethyl]-3-{[(4-fluorophenyl)methyl]amino}benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-[4-(difluoromethoxy)-2-methylphenyl]-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]quinoline-4-carboxylic acid
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
6-[(5-acetylthiophen-3-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
6-cyclopentyl-3-{[(3,3-dimethylcyclohexyl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
ethyl 1-[(3-methoxyphenyl)methyl]-5-(5-methyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-(2-methoxyethyl)-1-methyl-4-[(5-methylfuran-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
5-fluoro-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(3aS,7aR)-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
methyl 1-(2-methoxyethyl)-5-[(1-methoxypropan-2-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-fluorophenyl)ethan-1-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-oxoethyl}-1λ6-thiane-1,1-dione
4-(3,5-difluoro-4-methoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
1-cyclopentyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
5-[3-(1H-pyrazol-1-yl)phenyl]furan-2-carboxylic acid
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
{1-ethyl-5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-[(3R,4S)-4-(dimethylamino)-1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperidin-3-yl]propan-1-ol
1-(4-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperazin-1-yl)-3-methylbutan-1-one
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]acetic acid
2-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
1-[(3-fluorophenyl)methyl]-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(piperidin-1-yl)ethyl]acetamide
1,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(2,3-difluorophenoxymethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
1-{4-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1-cyclopentyl-N-[(2,3-dimethoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3-(1-methyl-1H-1,3-benzodiazol-6-yl)urea
N-ethyl-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
N-benzyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-[(3-ethenylphenyl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
N'-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-N,N-dimethylbutanediamide
6-fluoro-2-(1H-pyrazol-4-yl)-4-(thiomorpholine-4-carbonyl)quinoline
[4-(2-phenylethyl)-1-(quinoxalin-2-yl)piperidin-4-yl]methanol
N-[3-(1H-imidazol-1-yl)propyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
9-(2-methoxy-4-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one