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2-[5-(3-cyclohexyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyrazine
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
(3aR,6aR)-2-{[4-(2-hydroxyethoxy)phenyl]methyl}-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl](quinolin-2-ylmethyl)amine
1,7-dimethyl-N-[(1R,2S)-2-phenylcyclopropyl]-1H-indole-2-carboxamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
N-[2-(3-methoxyphenyl)-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
5-(1H-imidazol-1-ylmethyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]furan-2-carboxamide
(2E)-3-(1H-imidazol-4-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethan-1-one
N4-(isoquinolin-5-ylmethyl)-N4,6-dimethylpyrimidine-2,4-diamine
5-(6-aminopyridin-3-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)pyrimidin-2-amine
4-(1-ethylpiperidin-4-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[4-(3-{[(cyclopentylmethyl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
[4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-oxazepan-6-yl]methanol
(1R,3S)-3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}cyclopentane-1-carboxylic acid
4-(3,5-dimethyl-1-benzofuran-2-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
[5-(1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1H-imidazol-2-yl)furan-2-yl]methanol
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
1-(thiophene-2-carbonyl)-4-(2,4,5-trimethylbenzoyl)piperazine
N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)-4-(1H-pyrrol-1-yl)benzamide
1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
5-(4-methylphenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-4-amine
N-(3-{[methyl(1,3-thiazol-2-ylmethyl)carbamoyl]amino}phenyl)cyclopentanecarboxamide
8-(dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-4-carboxamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(pyridin-3-yl)propanamide
(furan-2-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(thiophen-3-ylmethyl)amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[3-(2-methylphenyl)phenyl]methyl}piperazine
(2S,4R)-N-methyl-4-{4-[(N-methyl-1-naphthalen-2-ylformamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
1-(3-acetylphenyl)-3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
6-(azepane-1-carbonyl)-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(4-ethoxy-3-methylphenyl)butan-1-one
7-{1-phenylspiro[2.4]heptane-1-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-4H-chromen-4-one
7-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indole
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1H-pyrazol-1-yl)ethyl]piperidin-2-one
1-(2-chlorophenyl)-3-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[4-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)phenyl]acetamide
N'-(2-ethoxyphenyl)-N-[(2-ethoxypyridin-3-yl)methyl]propanediamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]propan-1-one
1-(3-chlorophenyl)-3-{1,9-dioxaspiro[5.5]undecan-4-yl}urea
2-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-cyclopentyl-5-(2,3-difluoro-4-methoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole