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1-[(3-methoxyphenyl)methyl]-4-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]piperazin-2-one
(3R)-1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
(4aS,8aS)-N-(4-ethylphenyl)-4a-hydroxy-decahydroisoquinoline-2-carboxamide
1-(1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidin-4-yl)piperidine-3-carboxylic acid
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
9-[3-(1H-imidazol-1-yl)propyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
5-[6-(thiomorpholin-4-yl)pyridazin-3-yl]quinoline
N-(dimethyl-1H-1,2,4-triazol-5-yl)-3-{[(furan-3-ylmethyl)(methyl)amino]methyl}benzamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
2-{[4-(3-chlorophenyl)-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-chloro-N-(2-methoxyethyl)-4-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
3-(1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)benzoic acid
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]acetamide
3-methyl-5-[(phenylsulfanyl)methyl]-1H-1,2,4-triazole
3-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-[(4-methoxyphenyl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-methyl-6-oxo-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,6-dihydropyridazine-3-carboxamide
3-(azonan-1-yl)-N-(2,4-dimethylphenyl)-3-oxopropanamide
N-[(2-methoxyphenyl)methyl]-4,6-dimethylpyrimidin-2-amine
1-[(2-fluorophenyl)methyl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3-triazole-4-carboxamide
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-{5-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
2-[2-(furan-2-yl)-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetic acid
4-methyl-2-{2-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carboxamide
3-hydroxy-N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(2-methylphenyl)pyrrolidine-1-carboxamide
1-methyl-6-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,6-dihydropyridazine-3-carboxamide
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazole-2-carboxamide
3-ethyl-8-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-phenyl-1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidin-3-ol
3-hydroxy-3-({[2-(2-methylphenyl)ethyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-2-methylpyrimidine
2-{2-[1-(4-methylquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-benzyl-1-[2-(dimethylamino)ethyl]-3-[2-(methylsulfanyl)phenyl]urea
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-(2-methylpropyl)pyrimidine-5-carboxamide
N-[(2-chlorophenyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-{3-[(diethylamino)methyl]phenyl}-4-(morpholin-4-yl)piperidine-1-carboxamide
1-(9-methyl-9H-carbazole-3-carbonyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(2-fluorobenzenesulfonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(butan-2-yl)-N-(3-phenylprop-2-yn-1-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
4-[1-(naphthalene-1-sulfonyl)azetidin-3-yl]pyridine
N-(1H-indol-3-yl)pyridine-4-carboxamide
4-(4-fluorophenyl)-N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]piperazine-1-carboxamide
1-(4-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one