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N-[(3S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-(2-phenoxyethyl)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}urea
8-(4-methanesulfonylphenyl)-2-methylquinolin-4-ol
2-{1-[(2-methylphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{2-[(2-fluorophenyl)formamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-N-methylformamido}-N-methylbutanamide
(2-{[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)amino}ethyl)dimethylamine
2-(ethylamino)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
ethyl 4-[(benzylsulfamoyl)amino]piperidine-1-carboxylate
N-methyl-N-{3-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-3-oxopropyl}methanesulfonamide
1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(isoquinolin-1-yl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-(1-{1-[(5-acetamidoquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
(1R,5R)-3-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6-dimethoxypyridine
2-[2-(ethylsulfanyl)ethyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
N-(1H-imidazol-2-ylmethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-ethyl-3-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)piperidine
1-(3-benzoylpiperidin-1-yl)-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
2-hydroxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzoic acid
N-[2-(2,5-dimethylphenyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-ethyl-N-(1H-imidazol-2-ylmethyl)-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-[(3S,4R)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoate
(3R,4R)-4-(2-methoxyethyl)-1-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}-3-methylpiperidin-4-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,4-dioxane-2-carboxamide
(4aS,8aS)-2-[(3-tert-butyl-2-hydroxyphenyl)methyl]-decahydroisoquinolin-4a-ol
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-[(3S,4R)-1-benzyl-4-(morpholin-4-yl)piperidin-3-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
7-[1-(4-aminobutyl)-4-phenyl-1H-imidazol-5-yl]-2,6-dimethylheptan-2-ol
2-(5-ethylpyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
ethyl 3-[(6-hydroxy-1,4-oxazepane-4-carbonyl)amino]-6-methylthieno[2,3-b]pyridine-2-carboxylate
N-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}methanesulfonamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
4-[3-(azepane-1-carbonyl)-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-ethyl-3-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(3-ethyl-1H-pyrazol-5-yl)pyridine-3-carbonitrile
2-[3-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-1H-indol-1-yl]propanoic acid
2,3-dimethyl-5-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{4-[5-(aminomethyl)-2-fluorophenyl]phenyl}acetonitrile
2-cyclopropyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-N-tert-butylacetamide
2-amino-6-(4-chlorophenyl)-4-[5-(hydroxymethyl)furan-2-yl]-5-methylpyridine-3-carbonitrile
5-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]quinoline
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
5-chloro-7-methoxy-N-methyl-N-propyl-1-benzofuran-2-carboxamide
4-benzyl-3-ethyl-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,4-diazepan-5-one
N-cyclopropyl-5-(quinolin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide