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(2R,6S)-4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,6-dimethylmorpholine
3-(2-amino-1,3-thiazol-4-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
2-{4-[1-(3-methylfuran-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
4-cyclohexyl-3-oxo-N-(2-phenylphenyl)piperazine-1-carboxamide
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-methoxy-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-4-amine
1-(2-chlorophenyl)-4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazole
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3,5-dimethoxyphenyl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-{2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
N-[4-(furan-2-yl)butan-2-yl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[(1-{6-[(3S)-3-hydroxypyrrolidin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-N-(3-hydroxyphenyl)-4-oxobutanamide
9-(2,6-diaminopyrimidin-4-yl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-(6-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
N,8-dimethyl-N-[(5-methylfuran-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(oxan-4-yl)piperidine-3-carboxamide
5-[2-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]-2-methyl-3,4-dihydropyrimidin-4-one
pyridin-2-yl[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]methanol
4-(4-{[1-(4-chlorophenyl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
3-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
(3aS,6aS)-2-[3-(1H-imidazol-1-yl)propyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[ethyl(oxan-4-yl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
4-ethyl-N-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}cyclohexane-1-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(2,2,2-trifluoroethyl)acetamide
3,3,3-trifluoro-2-hydroxy-2-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}propanamide
N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-benzofuran-5-carboxamide
1-({5-[(3,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
8-fluoro-2-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoline
1-methyl-2-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
6-(2-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyridazin-3-amine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidine-1-carboxamide
N-methyl-1-({3-[(1-methyl-1H-pyrazol-4-yl)carbamoyl]phenyl}methyl)pyrrolidine-3-carboxamide
N-methyl-3-(3-methylpiperidin-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-(2-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-4-methyl-4H-1,2,4-triazole
3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-6-ethoxy-1,2-dihydroquinolin-2-one
6-[6-hydroxy-4-(3-hydroxy-1,2-oxazole-5-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
(1S,5R)-3-benzyl-6-(2,6-dimethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[4-(trifluoromethyl)phenyl]acetamide
(3R,4R)-4-cyclobutyl-3-methyl-1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]piperidin-4-ol
N3-{[4-(methylsulfanyl)phenyl]methyl}-N3-propylpiperidine-1,3-dicarboxamide
(2E)-N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,3-dihydro-1-benzofuran-7-carboxamide
2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
4-[(2-methylphenyl)methyl]-1-propyl-1,4-diazepan-5-one