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N-[1-(3-methylpyridin-2-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
1-(2,3-difluorobenzoyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
6-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile
3-ethoxy-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-cyclopropyl-4-({[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}methyl)pyrrolidin-2-one
methyl 3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}butanoate
4-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
N,N-dimethyl-2-[4-(1H-pyrazol-1-yl)phenyl]pyridine-3-carboxamide
9-[2-(dimethylamino)propanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-[5-(benzylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl]piperazine-1-carboxylate
2-(dimethylamino)-2-(4-methylphenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
(1R,2R,6S,7S)-4-[(1-benzyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-4-azatricyclo[5.2.1.02,6]decane
dimethyl({1-[4-(quinolin-3-yl)phenyl]ethyl})amine
(1S,5R)-3-[2-(3-chloro-4-hydroxyphenyl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-3-ol
7-[4-(1H-imidazol-1-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4'-(quinolin-8-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(2H-1,3-benzodioxol-5-yl)-2-[4-(4-ethylpiperazine-1-carbonyl)-5-(furan-2-yl)-1H-pyrazol-1-yl]pyrimidine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-[3-(2-methoxyphenyl)propyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
2-[4-(2,2-dimethylpropyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
8-[(1-methyl-1H-imidazol-5-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-{1-[4-methyl-4-(methylsulfanyl)pentan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N-[2-methyl-1-(pyridin-2-yl)propyl]-2-oxo-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
4-{1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}pyrimidine
N,N-diethyl-2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(3-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3,5-dimethyl-N-{3-methyl-1-[7-(oxolane-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
5-(methanesulfonylmethyl)-2-[3-(pyridin-4-yl)azetidin-1-yl]pyridine
N-cyclopropyl-2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
4-methyl-N-{1-[3-(methylsulfanyl)propanoyl]azepan-3-yl}-1,2,3-thiadiazole-5-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(6-methoxynaphthalene-2-carbonyl)piperidine
(2S,4S)-1-(4-chloro-2-fluorobenzoyl)-N-ethyl-4-propanamidopyrrolidine-2-carboxamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-propoxypiperidine
2-methyl-N-[3-(1H-pyrazol-3-yl)phenyl]propanamide
5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(2R)-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrrolidine-2-carboxamide
N-benzyl-5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 3-(2,6-dimethylpyrimidine-4-carbonyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-2-(2-oxoazepan-1-yl)-N-(quinolin-2-ylmethyl)acetamide
(3R)-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazine
1-benzyl-3-(2-methoxyethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione