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2-(4-acetylpiperazin-1-yl)-2-(2,3-difluorophenyl)acetic acid
2-(3-hydroxypropyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-propylphenyl)-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
5-amino-3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)furan-2-carboxamide
1-methyl-1'-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)benzamide
(1S,5R)-3-benzyl-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1H-imidazol-4-yl)ethyl]-4-[(oxolan-3-yl)sulfamoyl]benzamide
1-{2-[3-(4-chlorophenyl)piperidin-1-yl]-2-oxoethyl}-3-methylimidazolidin-2-one
5-({methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrimidin-2-amine
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[3-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-yl]methanol
3-[1-(4-cyano-1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
5-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
3-(2-fluoro-4-methoxyphenyl)-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-pyrazole
1-[4-(dimethylamino)azepan-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
N-[(3-methylthiophen-2-yl)methyl]-2-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]aniline
2-{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}pyridine
[2-methyl-2-(morpholin-4-yl)propyl][2-methyl-2-(morpholin-4-ylmethyl)propyl]amine
7-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(1-cycloheptyl-6-oxopiperidine-3-carbonyl)piperidine-4-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
3,4-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-4-(hydroxymethyl)piperidin-3-ol
2-(3-fluoropyridin-4-yl)-5-(methanesulfonylmethyl)pyridine
1-benzyl-2-methyl-1,4-diazepan-5-one
N-[2-(4-fluorophenyl)ethyl]-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]acetamide
4-benzyl-1-[(3-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperidine
2-[3-(2,2,2-trifluoroethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-(2,5-dimethoxyphenyl)-1-phenyl-1H-1,2,3,4-tetrazole
1-[(3,4-difluorophenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-ethyl-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-methylprop-2-en-1-yl)benzamide
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
5-methoxy-N-(2-methoxyethyl)-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
2-(2-methoxyethyl)-6-(1-methylpiperidin-4-yl)-3,4-dihydropyrimidin-4-one
N,N-dimethyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
(2,1,3-benzoxadiazol-5-ylmethyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine
2-chloro-5-acetamido-N-[2-methoxy-1-(pyridin-2-yl)ethyl]benzamide
3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1-(3-methanesulfonamidophenyl)urea
ethyl 4-{[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}piperidine-1-carboxylate
N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]propan-1-one
N-[(4-methoxypyridin-2-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
(4aR,8aS)-1-(cyclohexylmethyl)-6-(quinoxalin-6-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(2-chloro-6-methoxyphenyl)-4-(3,3,3-trifluoropropyl)pyrimidine
N,2-dicyclopropyl-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide