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1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxypropyl)piperidine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-acetamidobenzamide
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-4-yl)ethan-1-one
8-benzyl-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1,3-dihydroxy-2-methylpropan-2-yl)-1,3-oxazole-4-carboxamide
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(trifluoromethyl)sulfanyl]ethan-1-one
7-chloro-4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methylquinoline
(1R,5S)-8-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octane
1-{1-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]butan-2-yl}-4-methylpiperazine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-3-hydroxypyridine-2-carboxamide
2-{[cyclopropyl(1H-indol-5-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
4-methyl-6-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
5-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-(3-methylphenyl)pyridine-3-carbonitrile
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-propylpyridine-3-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(cyclopropylmethyl)amino]-5-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]benzamide
5,5-dimethyl-3-(2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-oxazolidine-2,4-dione
(3S,4S)-4-(pyrrolidin-1-yl)-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-3-ol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-indole-2-carboxamide
3-benzyl-4-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperazin-2-one
[1-(4-methylpyridine-3-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
3-[N-(2-phenylethyl)-1-1H-1,2,3-triazol-5-ylformamido]propanamide
2-(phenylsulfanyl)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
6-ethyl-N-methyl-2-(morpholin-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
3-(1-ethyl-1H-pyrazol-3-yl)-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
[(2-methoxyphenyl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amine
1,6-dimethyl-3-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-({1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(naphthalen-2-yl)piperazin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
6-ethyl-1,5-dimethyl-2-oxo-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
N-{[5-(2-ethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
2-methoxy-6-({3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)phenol
1-(furan-2-ylmethyl)-4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperazine
3-phenyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(1-methyl-1H-pyrazol-3-yl)-2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
5-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-{5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}-2-methylbutanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxybutanamide
4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one