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N-methyl-5-[({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)methyl]furan-2-carboxamide
1-(4-methylbenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
8-[(2-butyl-1H-imidazol-4-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-methoxyphenyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-2-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
2-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decane
3-[(2,6-dimethoxyphenyl)methyl]-5-methoxy-3,4-dihydroquinazolin-4-one
N-[3-(methylsulfanyl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine
1-(1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-(quinolin-6-yl)piperidine-1-carboxamide
2-(dimethylamino)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
(3aS,7aR)-5-methyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(3-methoxyphenyl)methyl]amine
4-[(4-fluorophenyl)methyl]-1-methylpiperidine
3-butyl-1-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)urea
2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
({4-[(6-methoxy-1-methyl-1H-indol-3-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
N,1-dimethyl-N-(oxan-2-ylmethyl)-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(4-methanesulfonylphenyl)pyrimidin-4-yl]piperidin-4-ol
N-cyclopropyl-5-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenyl-1,2-oxazole-4-carboxamide
2-(butan-2-ylsulfanyl)-5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidine
1-{2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]pyridine-4-carboxamide
(4aS,8aR)-6-(3,5-difluoropyridine-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(4aR,8aR)-2-(1H-indol-5-ylmethyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
4-[2-(dimethylamino)acetyl]-1-phenylpiperazin-2-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
5-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
1-[1'-(5-chloropyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(2S,4R)-4-amino-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N-methylpyrrolidine-2-carboxamide
4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
6-ethyl-2-methyl-N-[3-(3-oxopiperazin-1-yl)propyl]quinoline-4-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}carbamoyl)benzoate
4-(2-methyl-1-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-2-yl)morpholine
2-[1-cyclohexyl-4-(4-cyclopentylpyrimidin-2-yl)piperazin-2-yl]ethan-1-ol
1-{[3-(furan-2-yl)phenyl]methyl}-3-phenylpyrrolidin-3-ol
4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}phenol
1-[3-(azepane-1-carbonyl)benzenesulfonyl]-4-methyl-1,4-diazepane
N-{2-[(2-tert-butyl-4-hydroxypyrimidin-5-yl)formamido]ethyl}-2-chlorobenzamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
N-cyclooctyl-4-oxo-5-(piperidine-1-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(cyclohexylmethyl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1-(2-fluorophenyl)-4-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
3-({5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}methyl)-1λ6-thiolane-1,1-dione
2-[(3,5-difluorophenyl)methyl]-8-[(2S)-2,3-dihydroxypropyl]-2,8-diazaspiro[4.5]decan-3-one