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5-fluoro-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-4-(morpholin-4-yl)pyrimidin-2-amine
1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-(2-ethyl-1,3-dihydroxypropan-2-yl)-6-oxopiperidine-3-carboxamide
N,N-diethyl-3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(prop-2-en-1-yl)-1-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)urea
[(4-fluorophenyl)methyl](1H-imidazol-4-ylmethyl)(oxolan-2-ylmethyl)amine
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propylsulfanyl)ethan-1-one
2-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-{[4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine
4-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
2-tert-butyl-4-hydroxy-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}pyrimidine-5-carboxamide
2-methyl-6-(piperidin-4-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-4-amine
N-(1-ethyl-1H-indazol-3-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-1-(4-methoxyphenyl)piperazin-2-one
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidin-2-one
2-(azepan-1-yl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]acetamide
(1R,7S)-3-(2,2-dimethylpropyl)-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
[(3,7-dimethyl-1H-indol-2-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
ethyl 1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[3-(methylsulfanyl)propyl]urea
ethyl 1-ethyl-5-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-benzoyl-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidine
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl][2-(piperidin-1-yl)ethyl]amine
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
N-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2,3-difluorophenyl)ethan-1-one
2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[1-(2-methoxyphenyl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
3-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-[4-(2-methoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)acetamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}propanamide
(1S,2R)-2-[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]cyclohexan-1-ol
(3R,5R)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(naphthalen-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[2-(4-methoxyphenyl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-benzyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-[({1-[(2-chlorophenyl)methyl]-7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl}methyl)amino]-1λ6-thiolane-1,1-dione
4-methyl-1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)azepan-4-ol
N-benzyl-2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-sulfonamide
3,5-dimethyl-1-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-yl)-1H-pyrazole
2-(1-methyl-1H-pyrazole-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(cyclopropylmethyl)-7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1'-[(2,5-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-cyclohexyl-3-({[2-fluoro-6-(trifluoromethyl)phenyl]carbamoyl}amino)propanamide
methyl (2R,4S)-4-hydroxy-1-(5-propylthiophene-3-carbonyl)piperidine-2-carboxylate
2-[4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]pyrazine