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2-[5-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
9-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-6-methylpyridine-2-carboxamide
4-(benzyloxy)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
4-cyclobutyl-6-methyl-N-(oxolan-3-ylmethyl)pyrimidin-2-amine
ethyl 3-(2-methoxyethyl)-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoic acid
3-({1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidin-4-yl}oxy)pyridine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-benzothiophene-2-carboxamide
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-(pyrazin-2-yl)propan-1-one
2,3,5-trimethyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-2-propyl-3-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-(2-methoxyethyl)-1-{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2,6-dimethylquinoline-4-carboxamide
1-methyl-5-({4-oxo-6-propyl-3H,4H-thieno[2,3-d]pyrimidin-3-yl}methyl)pyrrolidin-2-one
4-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-3-fluoropyridine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
1-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-3-phenylpropan-1-one
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyridine
5-ethanesulfonamido-N,1-dimethyl-2-phenyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
2-(dimethylamino)-N-{[1-(ethoxymethyl)cyclopropyl]methyl}-2-(2-methylphenyl)acetamide
[4-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl](methyl)amino}methyl)oxan-4-yl]methanol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-3-oxopropanamide
N-({5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(naphthalen-2-yloxy)propan-1-one
5-{2-[4-(2-methoxynaphthalen-1-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine
2-(3-{1,4-diazabicyclo[3.2.2]nonan-4-ylmethyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-{2-methyl-1-[3-(pyrimidin-4-yl)piperidin-1-yl]propan-2-yl}morpholine
3-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.5]undecane
(3R,4S)-4-(5-methylfuran-2-yl)-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-amine
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(1H-pyrazol-1-yl)butanamide
ethyl 4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]piperidine-1-carboxylate
3-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-2,2-dimethylpropan-1-ol
3-{3-[6-(methoxycarbonyl)-1H-1,3-benzodiazol-2-yl]-1H-indol-1-yl}propanoic acid
N-(4-butoxyphenyl)-4-(furan-2-carbonyl)-1,4-diazepane-1-carboxamide
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N,2-dimethylthieno[2,3-d]pyrimidin-4-amine
1-(cyclopropylmethyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-butyl-5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
2,3-dimethyl-7-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}-1H-indole
N2-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
(2-phenylethyl)[(5,6,7-trimethoxy-2-phenylquinolin-3-yl)methyl]amine
5-(3-fluorophenoxymethyl)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazole
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
N-[(3S,4R)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-{6-methyl-5-[5-(2-phenylethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one