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3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]acetamide
4-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(2-chlorophenyl)-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
3-cyclohexyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
14-[(3Z)-hex-3-en-1-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
2,6-dimethyl-4-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}phenyl acetate
N,2-dimethyl-N-[2-(4-methylpiperidin-1-yl)ethyl]furan-3-carboxamide
2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
({5-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-cyano-N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-2-carboxamide
N-[2-(azepan-1-yl)ethyl]-3-methyl-N-(propan-2-yl)furan-2-carboxamide
2-(4-hydroxyphenyl)-N-[1-(piperidine-1-carbonyl)piperidin-4-yl]propanamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-ethyl-1-methylpiperazine
2-(5-methyl-1H-pyrazol-1-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
2,3-dimethyl-6-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoxaline
1-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
(2S)-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(cyclopropylmethyl)piperidine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-phenyl-4-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)-1,3-oxazole
3-(2-methoxyphenoxy)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}azetidine
9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-1-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[3-(2-methylphenyl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-[(prop-2-en-1-yl)amino]benzamide
N,4,6-trimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-2-amine
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
4-(azepan-1-yl)-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]propanamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propan-1-one
1-phenyl-2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethan-1-ol
2-(cyclohex-1-en-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(4aS,7aR)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-ethyl-1-methyl-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N3-(1-benzylpiperidin-4-yl)-1-(cyclohexylmethyl)-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[benzyl(methyl)amino]-3-(4-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
N-benzyl-3-oxo-2,8-diazaspiro[4.5]decane-8-sulfonamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-3-ylmethyl)amine
(1S,9S)-11-[6-(2-methoxyphenyl)pyridazin-3-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(pyridin-3-yl)ethyl]amine
1-{2-methoxy-4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
N-({1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}methyl)-4-phenylbenzamide
2-(1-tert-butyl-1H-pyrazol-4-yl)-4-(3-methylpiperidine-1-carbonyl)quinoline
cyclohexyl({4-[3-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide